SCHEMBL28102485

SCHEMBL28102485

Cc1cc(C(N)=O)cc(C)c1CC[C@H](NC(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 10/20 0.43
PPARG P37231 9/20 0.43
CTSK P43235 3/20 0.42
CTSS P25774 1/20 0.42
ACE P12821 1/20 0.42
PPARD Q03181 2/20 0.42
ITGB3 P05106 2/20 0.41
ITGA2B P08514 2/20 0.41
ITGB1 P05556 1/20 0.41
ITGAV P06756 1/20 0.41
ITGB5 P18084 1/20 0.41
ALDH1A1 P00352 1/20 0.40
TSHR P16473 1/20 0.40
IDO1 P14902 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19720147 1.00 PPARA (0.43) PPARAPPARGCTSKCTSSACE
SCHEMBL1055858 0.88 ACE (0.49) PPARAPPARGCTSKCTSSACE
SCHEMBL1055857 0.88 ACE (0.49) PPARAPPARGCTSKCTSSACE
SCHEMBL28102425 0.81 CTSK (0.48) PPARAPPARGCTSKCTSSACE
SCHEMBL28834742 0.81 CTSK (0.48) PPARAPPARGCTSKCTSSACE
SCHEMBL13316851 0.81 CTSS (0.40) PPARAPPARGCTSKCTSSACE
SCHEMBL1056766 0.80 KLK5 (0.45) PPARAPPARGCTSKCTSSACE
SCHEMBL1056763 0.80 KLK5 (0.45) PPARAPPARGCTSKCTSSACE
SCHEMBL12600964 0.79 ACE (0.42) PPARAPPARGCTSKCTSSACE
SCHEMBL16366761 0.78 ACE (0.49) PPARAPPARGCTSKCTSSACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102786476-B compounds as opioid receptor modulators 詹森药业有限公司 2017-01-18 CN disclosed