SCHEMBL28102787

SCHEMBL28102787

COc1ccc(Cn2ccc(C(C)C)c2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
MAPT P10636 2/20 0.45
KDM4E B2RXH2 1/20 0.45
ALOX15 P16050 1/20 0.45
CMA1 P23946 1/20 0.45
CYP19A1 P11511 1/20 0.45
NPBWR1 P48145 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.43
HSP90AA1 P07900 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
GSK3A P49840 1/20 0.42
GSK3B P49841 1/20 0.42
TP53 P04637 1/20 0.42
GAA P10253 1/20 0.42
SLC6A4 P31645 1/20 0.42
SIGMAR1 Q99720 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23920431 0.84 SIGMAR1 (0.49) ALDH1A1MAPTSMN1; SMN2NPC1RAB9A
SCHEMBL26202004 0.81 CYP19A1 (0.46) ALDH1A1MAPTCYP19A1SMN1; SMN2NPC1
SCHEMBL28170673 0.76 NPBWR1 (0.44) ALDH1A1MAPTKDM4EALOX15CMA1
SCHEMBL29709490 0.75 CYP19A1 (0.52) CMA1CYP19A1SMN1; SMN2HSP90AA1NPC1
SCHEMBL28321315 0.74 CA1 (0.53) ALDH1A1MAPTKDM4ECMA1CYP19A1
SCHEMBL11819451 0.73 MAPT (0.55) ALDH1A1MAPTKDM4EALOX15CMA1
SCHEMBL13975111 0.73 NPBWR1 (0.52) ALDH1A1MAPTKDM4EALOX15CMA1
SCHEMBL28434180 0.71 PTGS2 (0.53) ALDH1A1CMA1HSP90AA1GSK3AGSK3B
SCHEMBL28521022 0.70 CYP19A1 (0.45) ALDH1A1MAPTKDM4EALOX15CMA1
SCHEMBL1961673 0.70 CYP11B1 (0.49) ALDH1A1MAPTKDM4ECYP19A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106146484-A Quinazoline derivant is as RAF kinase modulator and their method and purposes 埃姆比特生物科学公司 2016-11-23 CN disclosed