SCHEMBL28104016

SCHEMBL28104016

CCNc1nc(Br)cnc1N

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 4/20 0.40
PGK1 P00558 2/20 0.37
EDNRA P25101 1/20 0.36
NUDT1 P36639 1/20 0.34
ATR Q13535 1/20 0.34
CCR4 P51679 3/20 0.33
KDM4E B2RXH2 1/20 0.33
NLRP3 Q96P20 1/20 0.33
MAPKAPK2 P49137 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12146478 0.82 ATR (0.35) NUDT1ATRCCR4HTTKMT2A
SCHEMBL15003295 0.78 PGK1 (0.45) PDE10APGK1EDNRACCR4KDM4E
SCHEMBL7322176 0.78 ADORA2A (0.37) EDNRAATRCCR4HTTKMT2A
SCHEMBL30588876 0.78 ADORA2A (0.37) EDNRAATRCCR4HTTKMT2A
SCHEMBL6825411 0.78 PDE10A (0.46) PDE10AMAPKAPK2HTT
SCHEMBL3018852 0.77 CRHR1 (0.38) ATRCCR4
SCHEMBL20387726 0.77 ALDH1A1 (0.44) ATRKDM4EL3MBTL1HTTKMT2A
SCHEMBL15803560 0.75 ATR (0.38) EDNRAATRCCR4HTTKMT2A
SCHEMBL20607670 0.74 TLR8 (0.47) EDNRAATRCCR4KMT2A
SCHEMBL21388100 0.74 ADORA3 (0.35) ATRCCR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102245611-B mTOR kinase inhibitors for use in mTOR/PI 3K/AKT/pathway-related oncology indications and diseases 西格诺药品有限公司 2016-10-26 CN disclosed