SCHEMBL28107018

SCHEMBL28107018

N#Cc1ccc2c(ccn2-c2cccnc2)c1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 5/20 0.56
CDC7 O00311 6/20 0.53
CYP11B2 P19099 5/20 0.50
CYP11B1 P15538 3/20 0.50
CYP17A1 P05093 1/20 0.50
PTGER2 P43116 1/20 0.49
ENPP3 O14638 1/20 0.47
CDK2 P24941 3/20 0.47
FFAR4 Q5NUL3 1/20 0.43
CHRNB2 P17787 1/20 0.41
CHRNA5 P30532 1/20 0.41
CHRNA4 P43681 1/20 0.41
MAP3K14 Q99558 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6654549 0.87 CYP11B2 (0.53) CYP19A1CDC7CYP11B2CYP11B1CYP17A1
SCHEMBL6663716 0.83 CYP11B2 (0.49) CYP19A1CDC7CYP11B2CYP11B1CYP17A1
SCHEMBL4282844 0.83 ENPP3 (0.56) CYP19A1CDC7ENPP3CDK2FFAR4
SCHEMBL6844281 0.82 CYP11B2 (0.57) CYP19A1CDC7CYP11B2CYP11B1CYP17A1
SCHEMBL15742146 0.81 CDC7 (0.51) CYP19A1CDC7CYP11B2PTGER2ENPP3
SCHEMBL3927305 0.80 PTGER2 (0.42) CYP19A1CDC7CYP11B2CYP11B1CYP17A1
SCHEMBL6658847 0.80 BRPF1 (0.60) CYP19A1
SCHEMBL28562388 0.78 CDC7 (0.60) CYP19A1CDC7CYP11B2CYP11B1CYP17A1
SCHEMBL17067754 0.78 ROCK1 (0.50) CYP19A1CYP11B2CYP11B1
SCHEMBL8306084 0.78 CYP19A1 (0.53) CYP19A1CYP11B2CYP11B1PTGER2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104193725-B Organic compound 诺华股份有限公司 2016-11-16 CN disclosed