SCHEMBL28111157

SCHEMBL28111157

CS(=O)(=O)C(c1ccccc1)c1cccc(-n2ccc(C(F)(F)F)c2)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.34
NR1H2 P55055 2/20 0.34
ACP3 P15309 1/20 0.33
PPARG P37231 2/20 0.33
DRD4 P21917 1/20 0.33
KDM4E B2RXH2 1/20 0.33
CASR P41180 1/20 0.33
COMT P21964 1/20 0.33
ACP1 P24666 1/20 0.32
PTPN7 P35236 1/20 0.32
PTPN12 Q05209 1/20 0.32
PTPN13 Q12923 1/20 0.32
SSU72 Q9NP77 1/20 0.32
LMNA P02545 2/20 0.32
KMT2A Q03164 1/20 0.32
PTGS2 P35354 2/20 0.32
TP53 P04637 1/20 0.32
MAPT P10636 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
G6PD P11413 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28111192 0.89 CASR (0.37) ACP3KDM4ECASRPTGS2
SCHEMBL28111761 0.75 IDO1 (0.47) ACP3PPARGDRD4KDM4ECASR
SCHEMBL31013537 0.73 ALDH1A1 (0.46) DRD4COMTLMNATP53MAPT
SCHEMBL28102822 0.71 HSP90AA1 (0.42) HTTKDM4EKMT2APTGS2ALDH1A1
SCHEMBL1272692 0.68 CYP2C19 (0.48) KDM4ELMNAKMT2AMAPTALDH1A1
SCHEMBL28121740 0.63 TSHR (0.52) HTTPTGS2MAPTALDH1A1
SCHEMBL28199860 0.61 CA2 (0.35) ALDH1A1
SCHEMBL22288889 0.61 HPGD (0.34) LMNAALDH1A1
SCHEMBL11937825 0.61 KDM4E (0.59) KDM4EALDH1A1
SCHEMBL14974088 0.59 ALDH1A1 (0.46) HTTKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106257976-A Human plasma kallikrein inhibitors 拜奥克里斯特制药公司 2016-12-28 CN disclosed