SCHEMBL28111761

SCHEMBL28111761

FC(F)(F)OC(c1ccccc1)c1cccc(-n2ccc(C(F)(F)F)c2)c1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 5/20 0.47
TDO2 P48775 5/20 0.47
DRD4 P21917 1/20 0.34
RXRA P19793 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2B Q13224 1/20 0.33
ACP3 P15309 1/20 0.32
PPARG P37231 2/20 0.32
CASR P41180 2/20 0.32
KDM4E B2RXH2 1/20 0.32
COMT P21964 1/20 0.32
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31013537 0.75 ALDH1A1 (0.46) DRD4COMTALDH1A1
SCHEMBL28111157 0.75 HTT (0.34) IDO1TDO2DRD4ACP3PPARG
SCHEMBL10654262 0.72 IDO1 (0.48) IDO1TDO2
SCHEMBL28102822 0.70 HSP90AA1 (0.42) KDM4EALDH1A1
SCHEMBL28111192 0.65 CASR (0.37) ACP3CASRKDM4E
SCHEMBL28199860 0.63 CA2 (0.35) ALDH1A1
SCHEMBL28121740 0.61 TSHR (0.52) ALDH1A1
SCHEMBL6140430 0.60 IDO1 (0.65) IDO1TDO2ACP3ALDH1A1
SCHEMBL28330130 0.60 MIF (0.41) RXRAGRIN1GRIN2B
SCHEMBL11937825 0.59 KDM4E (0.59) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106257976-A Human plasma kallikrein inhibitors 拜奥克里斯特制药公司 2016-12-28 CN disclosed