SCHEMBL28111192

SCHEMBL28111192

CS(=O)(=O)C(c1ccccc1)c1ccc(-n2ccc(C(F)(F)F)c2)cc1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CASR P41180 2/20 0.37
MCHR1 Q99705 10/20 0.36
KCNH2 Q12809 7/20 0.36
PTGS2 P35354 3/20 0.36
CYP3A4 P08684 4/20 0.35
ACP3 P15309 1/20 0.35
HSD11B1 P28845 1/20 0.34
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28111157 0.89 HTT (0.34) CASRPTGS2ACP3KDM4E
SCHEMBL31013537 0.76 ALDH1A1 (0.46) CYP3A4
SCHEMBL1272692 0.71 CYP2C19 (0.48) KDM4E
SCHEMBL28330130 0.67 MIF (0.41) MCHR1KCNH2PTGS2
SCHEMBL28111761 0.65 IDO1 (0.47) CASRACP3KDM4E
SCHEMBL28102822 0.62 HSP90AA1 (0.42) PTGS2CYP3A4KDM4E
SCHEMBL21216561 0.61 CA1 (0.38) CYP3A4ACP3CA1CA2CA9
SCHEMBL28199860 0.60 CA2 (0.35) MCHR1CA2
SCHEMBL11937825 0.60 KDM4E (0.59) KDM4E
SCHEMBL28111864 0.60 PKM (0.51) HSD11B1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106257976-A Human plasma kallikrein inhibitors 拜奥克里斯特制药公司 2016-12-28 CN disclosed