SCHEMBL28111318

SCHEMBL28111318

Nc1ccc(-c2n[nH]cc2N)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.42
ALDH1A1 P00352 3/20 0.42
TDP1 Q9NUW8 2/20 0.42
TP53 P04637 2/20 0.42
METAP2 P50579 1/20 0.39
KIT P10721 2/20 0.38
PDGFRB P09619 1/20 0.38
FGFR1 P11362 1/20 0.38
FGFR2 P21802 1/20 0.38
HSD17B10 Q99714 2/20 0.36
TAAR1 Q96RJ0 1/20 0.36
NPC1 O15118 3/20 0.35
RAB9A P51151 3/20 0.35
ASIC3 Q9UHC3 1/20 0.35
MEN1 O00255 4/20 0.35
KMT2A Q03164 4/20 0.35
MAPT P10636 3/20 0.35
BLM P54132 1/20 0.35
KDM4E B2RXH2 2/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27828569 0.83 MKNK1 (0.43) TP53METAP2NPC1RAB9AMEN1
SCHEMBL695299 0.83 METAP2 (0.37) ALDH1A1METAP2HSD17B10NPC1RAB9A
SCHEMBL2379590 0.83 ALOX15 (0.48) ALDH1A1HSD17B10NPC1RAB9AMEN1
SCHEMBL544500 0.83 ALOX15 (0.48) ALDH1A1HSD17B10NPC1RAB9AMEN1
SCHEMBL10775547 0.79 ALDH1A1 (0.39) CYP3A4ALDH1A1TDP1TP53METAP2
SCHEMBL6155891 0.79 PDE3B (0.39) CYP3A4ALDH1A1TDP1TP53METAP2
SCHEMBL22637221 0.79 SMN1; SMN2 (0.46) TDP1TP53METAP2PDGFRBTAAR1
SCHEMBL32670854 0.79 ALDH1A1 (0.39) ALDH1A1PDGFRBFGFR1FLT3
SCHEMBL27568104 0.77 ERBB2 (0.49) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL27875387 0.75 ADORA2A (0.38) ALDH1A1MAPTKDM4ESMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103717602-B Kinase inhibitors 加利福尼亚大学董事会 2016-11-09 CN disclosed