SCHEMBL28111319

SCHEMBL28111319

NC1(S(=O)(=O)c2ccc(F)cc2)CCC1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.47
PTGS1 P23219 3/20 0.47
RORC P51449 9/20 0.46
NR1I2 O75469 6/20 0.46
PSEN1 P49768 3/20 0.44
PSEN2 P49810 3/20 0.44
APH1B Q8WW43 3/20 0.44
NCSTN Q92542 3/20 0.44
APH1A Q96BI3 3/20 0.44
PSENEN Q9NZ42 3/20 0.44
EEF2K O00418 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28110706 0.96 RORC (0.49) PTGS2PTGS1RORCNR1I2PSEN1
SCHEMBL28111260 0.73 RORC (0.49) PTGS2RORCNR1I2PSEN1PSEN2
SCHEMBL28343237 0.72 RORC (0.48) PTGS2RORCNR1I2PSEN1PSEN2
SCHEMBL16877047 0.71 TRPA1 (0.41) PTGS2RORCNR1I2PSEN1PSEN2
SCHEMBL16880400 0.69 PHGDH (0.51) PTGS2RORCNR1I2
SCHEMBL13822796 0.68 ALDH1A1 (0.56) RORCNR1I2
SCHEMBL8643204 0.67 RORC (0.41) PTGS2PTGS1RORCNR1I2PSEN1
SCHEMBL13896735 0.67 ALDH1A1 (0.58) PTGS2PTGS1RORCNR1I2
SCHEMBL16232174 0.67 ALDH1A1 (0.55) RORCNR1I2PSEN1PSEN2APH1B
SCHEMBL5217170 0.67 MMP3 (0.50) PTGS2PTGS1RORCNR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106132931-B Carbocyclic ring sulfone ROR gamma modulators 百时美施贵宝公司 2019-08-02 CN disclosed
CN-106132931-A Carbocyclic ring sulfone ROR gamma modulators 百时美施贵宝公司 2016-11-16 CN disclosed