SCHEMBL28111669

SCHEMBL28111669

CS(=O)(=O)Nc1cccc(C(O)c2ccccc2F)c1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADRA2C P18825 1/20 0.52
ADRA1A P35348 1/20 0.52
ADRA1B P35368 1/20 0.52
ALDH1A1 P00352 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
KEAP1 Q14145 1/20 0.45
POLB P06746 1/20 0.43
NR3C1 P04150 2/20 0.43
KIF11 P52732 1/20 0.41
PGR P06401 1/20 0.40
NR3C2 P08235 1/20 0.40
AR P10275 1/20 0.40
HSD17B1 P14061 1/20 0.39
HSD17B2 P37059 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MAPKAPK2 P49137 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28111698 0.82 KEAP1 (0.58) ALDH1A1SMN1; SMN2KEAP1POLBNR3C1
SCHEMBL14677796 0.77 ALDH1A1 (0.44) ADRA2CADRA1AADRA1BALDH1A1SMN1; SMN2
SCHEMBL245468 0.76 MEN1 (0.60) ALDH1A1SMN1; SMN2KEAP1POLBHSD17B1
SCHEMBL229877 0.74 CES2 (0.45)
SCHEMBL28111139 0.73 ALDH1A1 (0.47) ADRA2CADRA1AADRA1BALDH1A1SMN1; SMN2
SCHEMBL31067420 0.72 IDO1 (0.42) ALDH1A1
SCHEMBL17064312 0.72 IDO1 (0.42) ALDH1A1
SCHEMBL10100499 0.72 KEAP1 (0.55) ALDH1A1SMN1; SMN2KEAP1POLBNR3C1
SCHEMBL7108854 0.72 ALDH1A1 (0.51) ADRA2CADRA1AADRA1BALDH1A1SMN1; SMN2
SCHEMBL13139256 0.72 ALDH1A1 (0.51) ADRA2CADRA1AADRA1BALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106257976-A Human plasma kallikrein inhibitors 拜奥克里斯特制药公司 2016-12-28 CN disclosed