SCHEMBL28111698

SCHEMBL28111698

CS(=O)(=O)Nc1cccc(C(O)c2ccccc2)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.58
ALDH1A1 P00352 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
POLB P06746 1/20 0.50
NR3C1 P04150 1/20 0.49
NR3C2 P08235 1/20 0.46
EGFR P00533 1/20 0.46
PIK3CA P42336 1/20 0.46
HSD17B1 P14061 1/20 0.44
HSD17B2 P37059 1/20 0.44
IKBKB O14920 1/20 0.44
CHUK O15111 1/20 0.44
USP2 O75604 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
TSHR P16473 1/20 0.44
CYP2C19 P33261 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28111139 0.83 ALDH1A1 (0.47) KEAP1ALDH1A1SMN1; SMN2POLBNR3C1
SCHEMBL245468 0.83 MEN1 (0.60) KEAP1ALDH1A1SMN1; SMN2POLBHSD17B1
SCHEMBL28111669 0.82 ADRA2C (0.52) KEAP1ALDH1A1SMN1; SMN2POLBNR3C1
SCHEMBL28111640 0.80 NPC1 (0.51) ALDH1A1SMN1; SMN2POLB
Diphenylmethanol SCHEMBL6670755 0.80 LMNA (0.55) KEAP1ALDH1A1SMN1; SMN2POLBCYP3A4
SCHEMBL10100499 0.79 KEAP1 (0.55) KEAP1ALDH1A1SMN1; SMN2POLBNR3C1
SCHEMBL17295589 0.79 TSHR (0.48) SMN1; SMN2EGFRPIK3CACYP3A4CYP2D6
SCHEMBL13139256 0.79 ALDH1A1 (0.51) KEAP1ALDH1A1SMN1; SMN2POLBNR3C1
SCHEMBL7108854 0.79 ALDH1A1 (0.51) KEAP1ALDH1A1SMN1; SMN2POLBNR3C1
SCHEMBL6500176 0.79 SMN1; SMN2 (0.55) KEAP1ALDH1A1SMN1; SMN2POLBNR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106257976-A Human plasma kallikrein inhibitors 拜奥克里斯特制药公司 2016-12-28 CN disclosed