SCHEMBL28111735

SCHEMBL28111735

O=C(NCC1CC1)c1ccc(Nc2cccc(Cl)c2)nn1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.56
CNR2 P34972 13/20 0.54
EPHX1 P07099 1/20 0.50
EPHX2 P34913 1/20 0.50
CYP3A4 P08684 4/20 0.48
CYP2C9 P11712 4/20 0.48
CYP2C19 P33261 4/20 0.48
CYP1A2 P05177 2/20 0.48
CYP2D6 P10635 2/20 0.48
DGAT1 O75907 1/20 0.48
NAMPT P43490 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28836629 0.81 VNN1 (0.56) CNR2DGAT1
SCHEMBL28111211 0.78 MT-CO2 (0.52) POLBCNR2CYP3A4CYP2C9CYP2C19
SCHEMBL28111270 0.78 CNR2 (0.60) POLBCNR2CYP3A4CYP2C9CYP2C19
SCHEMBL938902 0.75 NAMPT (0.47) NAMPT
SCHEMBL5214258 0.74 CNR2 (0.91) CNR2CYP3A4CYP2C9CYP2C19CYP1A2
SCHEMBL5214314 0.74 CNR2 (0.75) CNR2EPHX1EPHX2CYP3A4CYP2C9
SCHEMBL5212538 0.74 CNR2 (0.93) CNR2CYP3A4CYP2C9CYP2C19CYP1A2
SCHEMBL5212134 0.74 CNR2 (0.75) CNR2EPHX1EPHX2CYP3A4CYP2C9
SCHEMBL5214918 0.73 CNR2 (0.69) POLBCNR2EPHX1EPHX2CYP3A4
SCHEMBL5216408 0.73 CNR2 (0.75) CNR2EPHX1EPHX2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106187910-A Pyridazine class derivant and its production and use 浙江大学 2016-12-07 CN claimed
CN-106187910-A Pyridazine class derivant and its production and use 浙江大学 2016-12-07 CN disclosed