SCHEMBL28111270

SCHEMBL28111270

O=C(NCc1ccc(F)cc1)c1ccc(Nc2cccc(Cl)c2)nn1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 8/20 0.60
RAB9A P51151 1/20 0.58
CYP1A2 P05177 2/20 0.55
CYP2C9 P11712 2/20 0.55
CYP2C19 P33261 2/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2D6 P10635 1/20 0.55
ALDH1A1 P00352 2/20 0.52
MEN1 O00255 1/20 0.52
LMNA P02545 1/20 0.52
MAPT P10636 1/20 0.52
MAOA P21397 1/20 0.52
MAOB P27338 1/20 0.52
KMT2A Q03164 1/20 0.52
MT-CO2 P00403 1/20 0.52
TP53 P04637 2/20 0.48
POLB P06746 1/20 0.48
DGAT1 O75907 1/20 0.46
VNN1 O95497 1/20 0.45
MTOR P42345 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28836629 0.90 VNN1 (0.56) CNR2RAB9AMEN1LMNAMAPT
SCHEMBL28111211 0.89 MT-CO2 (0.52) CNR2RAB9ACYP1A2CYP2C9CYP2C19
SCHEMBL28111735 0.78 POLB (0.56) CNR2CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL28111733 0.77 MMP13 (0.52) CNR2RAB9ACYP1A2CYP2C19CYP2D6
SCHEMBL28111776 0.77 MAPT (0.64) CNR2CYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL5459863 0.76 CNR2 (0.81) CNR2RAB9ACYP1A2CYP2C9CYP2C19
SCHEMBL5078904 0.75 CNR2 (1.00) CNR2RAB9ACYP1A2CYP2C9CYP2C19
SCHEMBL6379713 0.71 TP53 (0.57) RAB9ACYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL5083343 0.71 CNR2 (1.00) CNR2CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL5457653 0.70 CNR2 (0.74) CNR2CYP1A2CYP2C9CYP2C19CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106187910-A Pyridazine class derivant and its production and use 浙江大学 2016-12-07 CN claimed
CN-106187910-A Pyridazine class derivant and its production and use 浙江大学 2016-12-07 CN disclosed