SCHEMBL28112786

SCHEMBL28112786

O=C1c2ncc(-c3cccc(Br)c3)cc2-c2cc(-c3cccc(Br)c3)cnc21

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BIRC5 O15392 1/20 0.51
MAOB P27338 1/20 0.47
GABRG2 P18507 9/20 0.44
GABRB3 P28472 9/20 0.44
GABRA5 P31644 9/20 0.44
GABRA3 P34903 9/20 0.44
GABRA1 P14867 7/20 0.44
IDO1 P14902 2/20 0.40
TDP2 O95551 1/20 0.39
METAP2 P50579 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
HRH1 P35367 1/20 0.38
HRH4 Q9H3N8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28112338 0.81 NPC1 (0.42) MAOBTDP2MEN1KMT2A
SCHEMBL28112787 0.72 DYRK1A (0.39) TDP2MEN1KMT2A
SCHEMBL29546450 0.71 ALDH1A1 (0.52) BIRC5MAOBGABRG2GABRB3GABRA5
SCHEMBL312091 0.71 ALDH1A1 (0.52) BIRC5MAOBGABRG2GABRB3GABRA5
SCHEMBL17460460 0.70 GABRG2 (0.55) BIRC5GABRG2GABRB3GABRA5GABRA3
SCHEMBL16601738 0.70 MAP4K4 (0.56) MEN1
SCHEMBL12441009 0.69 BIRC5 (0.54) BIRC5GABRG2GABRB3GABRA5GABRA3
SCHEMBL12556925 0.69 NPC1 (0.50) MAOBTDP2MEN1KMT2A
SCHEMBL29398919 0.69 ALDH1A1 (0.50) BIRC5MAOBGABRG2GABRB3GABRA5
SCHEMBL191276 0.69 ALDH1A1 (0.50) BIRC5MAOBGABRG2GABRB3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106188037-A A kind of compound based on 1,8-diaza-9-Fluorenone and application thereof 中节能万润股份有限公司 2016-12-07 CN disclosed