SCHEMBL28114119

SCHEMBL28114119

O=C(NC1(c2ccccc2C(F)(F)F)CC1)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.55
HDAC6 Q9UBN7 2/20 0.55
HDAC3 O15379 1/20 0.55
HDAC2 Q92769 1/20 0.55
HDAC4 P56524 1/20 0.50
KCNK3 O14649 1/20 0.44
KCNK9 Q9NPC2 1/20 0.44
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
LMNA P02545 2/20 0.42
MEN1 O00255 1/20 0.42
MAPT P10636 1/20 0.42
KMT2A Q03164 1/20 0.42
FAAH O00519 1/20 0.41
GAA P10253 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HSD17B10 Q99714 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
POLB P06746 1/20 0.40
TRPV1 Q8NER1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28113612 0.78 PDE2A (0.58) HDAC1HDAC6HDAC3HDAC2NPC1
SCHEMBL25375689 0.75 HDAC6 (0.48) HDAC1HDAC6HDAC3HDAC2HDAC4
SCHEMBL28793250 0.74 CXCR3 (0.51) HDAC1HDAC6HDAC3HDAC2LMNA
SCHEMBL4729552 0.71 HDAC3 (1.00) HDAC1HDAC6HDAC3HDAC2HDAC4
SCHEMBL23777401 0.71 NPC1 (0.50) HDAC1HDAC6HDAC3HDAC2NPC1
SCHEMBL4555610 0.71 HDAC4 (0.62) HDAC1HDAC6HDAC3HDAC2HDAC4
SCHEMBL19469572 0.70 HDAC4 (0.65) HDAC1HDAC6HDAC3HDAC2HDAC4
SCHEMBL30008296 0.68 POLB (0.67) HDAC1HDAC6HDAC3HDAC2KCNK3
SCHEMBL10605790 0.68 LMNA (0.51) HDAC1HDAC6HDAC3HDAC2LMNA
SCHEMBL6170575 0.68 POLB (0.67) HDAC1HDAC6HDAC3HDAC2KCNK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104487433-B Triazolone compounds as mPGES-1 inhibitors 格兰马克药品股份有限公司 2016-12-07 CN disclosed