SCHEMBL28113612

SCHEMBL28113612

O=C(NC1(c2ccc(C(F)(F)F)cc2)CC1)c1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 9/20 0.58
PTGER4 P35408 5/20 0.54
NPC1 O15118 1/20 0.54
RAB9A P51151 1/20 0.54
HDAC3 O15379 1/20 0.52
HDAC1 Q13547 1/20 0.52
HDAC2 Q92769 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
PTGER2 P43116 2/20 0.52
TBXA2R P21731 1/20 0.51
PTGER1 P34995 1/20 0.51
PTGFR P43088 1/20 0.51
PTGER3 P43115 1/20 0.51
PTGDR Q13258 1/20 0.51
KDM4E B2RXH2 1/20 0.50
APAF1 O14727 1/20 0.50
TDP2 O95551 1/20 0.50
NSD2 O96028 1/20 0.50
MAPT P10636 1/20 0.50
CASP3 P42574 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28793250 0.85 CXCR3 (0.51) HDAC3HDAC1HDAC2HDAC6KDM4E
SCHEMBL27075244 0.84 PDE2A (0.54) PDE2APTGER4HDAC3HDAC1HDAC2
SCHEMBL19282949 0.80 PDE2A (0.51) PDE2APTGER4HDAC3HDAC1HDAC2
SCHEMBL10605790 0.79 LMNA (0.51) PDE2AHDAC3HDAC1HDAC2HDAC6
SCHEMBL28114119 0.78 HDAC1 (0.55) NPC1RAB9AHDAC3HDAC1HDAC2
SCHEMBL23796172 0.77 PDE2A (0.48) PDE2APTGER4HDAC6PTGER2TBXA2R
SCHEMBL30290147 0.77 PDE2A (0.48) PDE2APTGER4HDAC6PTGER2TBXA2R
SCHEMBL15021087 0.76 SLC6A9 (0.79)
SCHEMBL16249346 0.76 WDR91 (0.53) PDE2AHDAC3HDAC1HDAC2HDAC6
SCHEMBL9188439 0.75 SLC6A9 (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104487433-B Triazolone compounds as mPGES-1 inhibitors 格兰马克药品股份有限公司 2016-12-07 CN disclosed