SCHEMBL28114866

SCHEMBL28114866

CCc1cc(C(=O)OC)cc2ccn(Cl)c12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.39
ALDH1A1 P00352 4/20 0.39
LMNA P02545 3/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
PTPN11 Q06124 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
HPGD P15428 2/20 0.39
HSD17B10 Q99714 2/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.39
ALOX15 P16050 1/20 0.39
ALOX12 P18054 1/20 0.39
APEX1 P27695 1/20 0.39
CASP1 P29466 1/20 0.39
RECQL P46063 1/20 0.39
BLM P54132 1/20 0.39
CASP7 P55210 1/20 0.39
RXFP1 Q9HBX9 1/20 0.38
CA12 O43570 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28114808 0.84 PTPN11 (0.36) KDM4EALDH1A1MEN1KMT2APTPN11
SCHEMBL28025056 0.84 ALDH1A1 (0.39) KDM4EALDH1A1MEN1KMT2APTPN11
SCHEMBL28025606 0.79 ALDH1A1 (0.40) KDM4EALDH1A1LMNAMEN1KMT2A
SCHEMBL8922937 0.77 CYP3A4 (0.43) KDM4EALDH1A1LMNAMEN1KMT2A
SCHEMBL28114800 0.73 KDM4E (0.48) KDM4EALDH1A1LMNAMEN1KMT2A
SCHEMBL28025597 0.72 ALDH1A1 (0.34) KDM4EALDH1A1CA12CA1CA2
SCHEMBL28025040 0.70 FBP1 (0.36) KDM4EALDH1A1LMNAMEN1KMT2A
SCHEMBL12419947 0.70 HPGD (0.48) KDM4EALDH1A1LMNAMEN1KMT2A
SCHEMBL22489748 0.70 KDM4E (0.54) KDM4EALDH1A1LMNAMEN1KMT2A
SCHEMBL29136490 0.69 CA1 (0.52) KDM4EALDH1A1LMNATDP1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104854087-B Indole carboxamide derivatives as P2X receptor antagonists 埃科特莱茵药品有限公司 2017-03-22 CN disclosed
CN-104812749-B Indolecarboxamide derivant as P2X7 receptor antagonist 埃科特莱茵药品有限公司 2016-12-14 CN disclosed