SCHEMBL28115901

SCHEMBL28115901

[CH2]CCNC(=O)c1cc(F)cc(C(F)(F)F)c1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RHOC P08134 5/20 0.48
RHOA P61586 5/20 0.48
DDR1 Q08345 1/20 0.47
ALDH1A1 P00352 1/20 0.47
POLB P06746 1/20 0.47
TACR1 P25103 1/20 0.46
RXFP1 Q9HBX9 1/20 0.43
MLYCD O95822 1/20 0.43
TP53BP1 Q12888 1/20 0.42
VNN1 O95497 2/20 0.41
GAA P10253 1/20 0.41
CES2 O00748 1/20 0.41
NNMT P40261 1/20 0.40
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28000419 0.91 RHOC (0.52) RHOCRHOADDR1ALDH1A1POLB
SCHEMBL13753113 0.85 ALDH1A1 (0.65) RHOCRHOADDR1ALDH1A1POLB
SCHEMBL13753001 0.81 DDR1 (0.55) RHOCRHOADDR1ALDH1A1POLB
SCHEMBL615458 0.80 TACR1 (0.50) RHOCRHOADDR1TACR1MLYCD
SCHEMBL14528862 0.79 RHOC (0.48) RHOCRHOADDR1ALDH1A1POLB
SCHEMBL27791536 0.77 MEN1 (0.63) ALDH1A1HDAC3HDAC1HDAC2HDAC6
Hydrochloric Acid SCHEMBL27791610 0.76 MEN1 (0.62) ALDH1A1POLB
SCHEMBL14214023 0.76 CES2 (0.47) DDR1TACR1RXFP1VNN1GAA
SCHEMBL25757925 0.76 CES2 (0.47) RHOCRHOADDR1TACR1VNN1
SCHEMBL14430729 0.75 KMT2A (0.54) RHOCRHOAALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104496962-B A kind of Oligopoly thiophene derivative and application thereof 南方医科大学 2017-01-04 CN disclosed
CN-104496962-A Oligothiophene derivative and application thereof UNIV SOUTHERN MEDICAL 2015-04-08 CN disclosed