SCHEMBL28115964

SCHEMBL28115964

COc1ccc(CN2CN(c3ccccc3)C=N2)cc1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.50
CYP11B1 P15538 1/20 0.48
CYP11B2 P19099 1/20 0.48
LTA4H P09960 1/20 0.42
LMNA P02545 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
NPBWR1 P48145 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14764819 0.72 DRD2 (0.51) SIGMAR1LMNAMAPTKMT2AL3MBTL1
SCHEMBL28115619 0.70 MAPT (0.43) SIGMAR1LMNAMAPTKMT2AALDH1A1
SCHEMBL14764534 0.69 DRD2 (0.53) SIGMAR1LMNAMAPTKMT2AL3MBTL1
SCHEMBL31548632 0.68 NPC1 (0.33) NPC1RAB9A
SCHEMBL28115961 0.67 ALDH1A1 (0.41) LMNAKDM4EMAPTKMT2AALDH1A1
SCHEMBL30579890 0.67 SIGMAR1 (0.47) SIGMAR1LMNAKDM4EMAPTKMT2A
SCHEMBL6450318 0.66 SIGMAR1 (0.67) SIGMAR1LMNAKDM4EMAPTALDH1A1
SCHEMBL1950743 0.65 CYP11B1 (1.00) SIGMAR1CYP11B1CYP11B2
SCHEMBL1548440 0.64 SIGMAR1 (0.50) SIGMAR1LTA4HKDM4EMAPTKMT2A
SCHEMBL15429645 0.63 CMA1 (0.58) SIGMAR1LMNAKDM4EMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106234385-B A kind of application of 1,2,4- triazole derivatives of the structure containing benzopyrazines as fungicide 浙江工业大学 2018-11-13 CN disclosed
CN-106432245-B A kind of 1,2,4- triazole derivatives of the structure containing benzopyrazines and its preparation method and application 浙江工业大学 2018-11-13 CN disclosed
CN-106432245-A 1,2,4-triazole derivative having quinoxaline structure, preparation method and application thereof 浙江工业大学 2017-02-22 CN disclosed
CN-106234385-A A kind of 1,2,4 triazole derivatives containing benzopyrazines structure are as the application of antibacterial 浙江工业大学 2016-12-21 CN disclosed