SCHEMBL28115994

SCHEMBL28115994

Oc1ncncc1-c1cccs1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 9/20 0.42
CYP2C9 P11712 7/20 0.42
CYP2E1 P05181 1/20 0.42
CYP2A6 P11509 1/20 0.42
CYP2B6 P20813 1/20 0.42
TDO2 P48775 1/20 0.41
ALDH1A1 P00352 9/20 0.40
CYP1A2 P05177 8/20 0.40
HSD17B10 Q99714 6/20 0.40
MEN1 O00255 5/20 0.40
KMT2A Q03164 5/20 0.40
CASP1 P29466 5/20 0.40
CASP7 P55210 5/20 0.40
USP2 O75604 4/20 0.40
CLK4 Q9HAZ1 3/20 0.40
HIF1A Q16665 1/20 0.40
CYP2C19 P33261 5/20 0.39
CYP2D6 P10635 4/20 0.39
TSHR P16473 4/20 0.39
MAPK1 P28482 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31452802 0.75 CYP3A4 (0.46) CYP3A4CYP2C9CYP2E1CYP2A6CYP2B6
SCHEMBL15660874 0.71 ADRB1 (0.43) CYP3A4CYP2C9CYP2E1CYP2A6CYP2B6
SCHEMBL7128234 0.70 TOP2A (0.38) TDO2ALDH1A1MEN1KMT2ACLK4
SCHEMBL16968469 0.69 CDK8 (0.59) CYP3A4CYP2C9CYP2E1CYP2A6CYP2B6
SCHEMBL219003 0.69 CYP3A4 (0.45) CYP3A4CYP2C9CYP2E1CYP2A6CYP2B6
SCHEMBL18789395 0.69 CYP3A4 (0.67) CYP3A4CYP2C9CYP2E1CYP2A6CYP2B6
SCHEMBL9438562 0.68 ALDH1A1 (0.46) CYP3A4CYP2C9CYP2E1CYP2A6CYP2B6
SCHEMBL14027112 0.68 RPS6KB2 (0.53) TDO2ALDH1A1HSD17B10MEN1KMT2A
SCHEMBL18133656 0.68 ERN1 (0.50) TDO2ALDH1A1HSD17B10MEN1KMT2A
SCHEMBL28423248 0.67 CYP3A4 (0.44) CYP3A4CYP2C9CYP2E1CYP2A6CYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106117194-A Can be used as 2 benzyls of SGC stimulant, 3 (pyrimidine 2 base) substituted pyrazoles 铁木医药有限公司 2016-11-16 CN disclosed