SCHEMBL28116823

SCHEMBL28116823

O=C(O)C1CCN(Cc2cccc(Oc3ccccc3)c2)C1=O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR8 P51685 4/20 0.53
KDM4E B2RXH2 4/20 0.51
ALDH1A1 P00352 3/20 0.51
LMNA P02545 1/20 0.51
GAA P10253 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
F10 P00742 1/20 0.48
FAAH O00519 2/20 0.48
TDP1 Q9NUW8 1/20 0.48
HPGD P15428 1/20 0.48
HTT P42858 1/20 0.48
APP P05067 2/20 0.47
MMP1 P03956 1/20 0.47
MMP2 P08253 1/20 0.47
MMP7 P09237 1/20 0.47
MMP10 P09238 1/20 0.47
MMP9 P14780 1/20 0.47
MMP13 P45452 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28116468 0.93 CCR8 (0.51) CCR8KDM4EALDH1A1LMNAGAA
SCHEMBL17048430 0.87 CCR8 (0.66) CCR8KDM4EALDH1A1LMNAGAA
SCHEMBL892946 0.84 HDAC1 (0.51) ALDH1A1GAAMEN1KMT2APOLB
SCHEMBL27491805 0.84 HDAC1 (0.51) ALDH1A1GAAMEN1KMT2APOLB
SCHEMBL4349231 0.83 KMT2A (0.53) CCR8KDM4EALDH1A1LMNAGAA
SCHEMBL17099382 0.82 KDM4E (0.50) CCR8KDM4EALDH1A1LMNAGAA
SCHEMBL17048461 0.80 CCR8 (0.63) CCR8KDM4EALDH1A1LMNAMEN1
SCHEMBL28961034 0.78 KMT2A (0.53) KDM4EALDH1A1MEN1KMT2APOLB
SCHEMBL4349232 0.77 MEN1 (0.51) CCR8KDM4EALDH1A1LMNAGAA
SCHEMBL5369178 0.76 L3MBTL1 (0.49) ALDH1A1GAAMEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106255679-B As NAThe heterocyclic compound and application thereof of V channel inhibitor 默克专利有限公司 2019-09-06 CN disclosed
CN-106255679-A As Naheterocyclic compound of V channel inhibitor and application thereof 默克专利有限公司 2016-12-21 CN disclosed