SCHEMBL28116468

SCHEMBL28116468

O=C(O)C1CCCN(Cc2cccc(Oc3ccccc3)c2)C1=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR8 P51685 4/20 0.51
KDM4E B2RXH2 4/20 0.51
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
APP P05067 3/20 0.49
MMP1 P03956 1/20 0.49
MMP2 P08253 1/20 0.49
MMP7 P09237 1/20 0.49
MMP10 P09238 1/20 0.49
MMP9 P14780 1/20 0.49
MMP13 P45452 1/20 0.49
PSEN1 P49768 1/20 0.49
PSEN2 P49810 1/20 0.49
MMP14 P50281 1/20 0.49
ADAM17 P78536 1/20 0.49
APH1B Q8WW43 1/20 0.49
NCSTN Q92542 1/20 0.49
APH1A Q96BI3 1/20 0.49
PSENEN Q9NZ42 1/20 0.49
ALDH1A1 P00352 3/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28116823 0.93 CCR8 (0.53) CCR8KDM4EMEN1KMT2AAPP
SCHEMBL4349231 0.88 KMT2A (0.53) CCR8KDM4EMEN1KMT2AAPP
SCHEMBL17048461 0.87 CCR8 (0.63) CCR8KDM4EMEN1KMT2AAPP
SCHEMBL5369178 0.85 L3MBTL1 (0.49) MEN1KMT2AALDH1A1GAA
SCHEMBL9740346 0.81 L3MBTL1 (0.51) MEN1KMT2AAPPALDH1A1GAA
SCHEMBL17048430 0.80 CCR8 (0.66) CCR8KDM4EMEN1KMT2AAPP
SCHEMBL4349232 0.80 MEN1 (0.51) CCR8KDM4EMEN1KMT2AAPP
SCHEMBL9205385 0.80 L3MBTL1 (0.54) MEN1KMT2AAPPALDH1A1
SCHEMBL17099382 0.78 KDM4E (0.50) CCR8KDM4EMEN1KMT2AAPP
SCHEMBL892946 0.77 HDAC1 (0.51) MEN1KMT2AALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106255679-B As NAThe heterocyclic compound and application thereof of V channel inhibitor 默克专利有限公司 2019-09-06 CN disclosed
CN-106255679-A As Naheterocyclic compound of V channel inhibitor and application thereof 默克专利有限公司 2016-12-21 CN disclosed