SCHEMBL28117528

SCHEMBL28117528

COc1ccc(-c2csc(Nc3cc(OC)c(OC)c(OC)c3)n2)cc1OC

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 2/20 0.69
CYP1A2 P05177 2/20 0.69
CYP1B1 Q16678 2/20 0.69
ALOX5 P09917 1/20 0.67
MEN1 O00255 11/20 0.67
KMT2A Q03164 11/20 0.67
MAPT P10636 5/20 0.67
POLB P06746 1/20 0.64
RAB9A P51151 6/20 0.63
NPC1 O15118 5/20 0.63
MAPK1 P28482 2/20 0.63
HTT P42858 1/20 0.63
GAA P10253 3/20 0.62
ALDH1A1 P00352 2/20 0.62
ALOX15 P16050 1/20 0.62
HSD17B10 Q99714 1/20 0.62
SMN1; SMN2 Q16637 2/20 0.61
PTGS2 P35354 2/20 0.56
PTGES O14684 1/20 0.55
PLAU P00749 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28117517 0.90 PTGES (0.68) CYP1A1CYP1A2CYP1B1ALOX5MEN1
SCHEMBL28117525 0.90 MEN1 (0.59) CYP1A1CYP1A2CYP1B1ALOX5MEN1
SCHEMBL28117523 0.90 ALOX5 (0.59) CYP1A1CYP1A2CYP1B1ALOX5MEN1
SCHEMBL28330115 0.88 PTGS2 (0.73) CYP1A1CYP1A2CYP1B1ALOX5MEN1
SCHEMBL12298237 0.88 MEN1 (0.65) CYP1A1CYP1A2CYP1B1ALOX5MEN1
SCHEMBL14458591 0.88 ALOX5 (0.62) CYP1A1CYP1A2CYP1B1ALOX5MEN1
SCHEMBL28117072 0.88 MEN1 (0.64) CYP1A1CYP1A2CYP1B1ALOX5MEN1
SCHEMBL12298231 0.87 CYP1B1 (0.67) CYP1A1CYP1A2CYP1B1ALOX5MEN1
SCHEMBL12297793 0.87 ALOX5 (0.61) CYP1A1CYP1A2CYP1B1ALOX5MEN1
SCHEMBL1890637 0.87 BRAF (0.62) CYP1A1CYP1A2CYP1B1ALOX5MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106220582-B n, 4-diaryl thiazole-2-amine compound and application thereof as tumor cell proliferation inhibitor 沈阳药科大学 2019-12-10 CN claimed
CN-106220582-A N, 4 diaryl thiazole 2 aminated compoundss and the purposes as tumor cell proliferation inhibitor thereof 沈阳药科大学 2016-12-14 CN claimed
CN-106220582-B n, 4-diaryl thiazole-2-amine compound and application thereof as tumor cell proliferation inhibitor 沈阳药科大学 2019-12-10 CN disclosed
CN-106220582-A N, 4 diaryl thiazole 2 aminated compoundss and the purposes as tumor cell proliferation inhibitor thereof 沈阳药科大学 2016-12-14 CN disclosed