SCHEMBL28118833

SCHEMBL28118833

O=C1Nc2ccc(Nc3ccc(F)cc3)cc2C1(O)Cc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.47
GSK3B P49841 2/20 0.43
NQO2 P16083 1/20 0.42
TP53 P04637 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
PGR P06401 1/20 0.38
HTT P42858 2/20 0.38
BRD4 O60885 1/20 0.37
PIK3CD O00329 1/20 0.37
MEN1 O00255 1/20 0.36
POLB P06746 1/20 0.36
KMT2A Q03164 1/20 0.36
IDO1 P14902 3/20 0.36
TDO2 P48775 1/20 0.36
PDK2 Q15119 1/20 0.36
MAPT P10636 2/20 0.36
EPHX2 P34913 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28119211 0.88 IDO1 (0.47) ATMGSK3BNQO2TP53SMN1; SMN2
SCHEMBL28119199 0.83 KIF11 (0.50) ATMHTTMEN1KMT2AMAPT
SCHEMBL28837904 0.79 NQO2 (0.47) GSK3BNQO2SMN1; SMN2BRD4MEN1
SCHEMBL28119198 0.79 NQO2 (0.47) GSK3BNQO2HTTBRD4MEN1
SCHEMBL28119197 0.78 NQO2 (0.46) GSK3BNQO2HTTBRD4MEN1
SCHEMBL2495439 0.76 IDO1 (0.62) ATMTP53SMN1; SMN2PGRPIK3CD
SCHEMBL17166881 0.76 ATM (0.55) ATMGSK3BTP53SMN1; SMN2PGR
SCHEMBL15426102 0.76 TP53 (0.67) ATMTP53SMN1; SMN2PGRPIK3CD
SCHEMBL12165522 0.74 ATM (0.77) ATMSMN1; SMN2HTTMEN1KMT2A
SCHEMBL28874851 0.70 KCNH3 (0.39) TP53MEN1POLBKMT2APDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106316923-A Disubstituted indol-2(1H)-one derivative and preparation method and application thereof 中南大学 2017-01-11 CN claimed
CN-106316923-A Disubstituted indol-2(1H)-one derivative and preparation method and application thereof 中南大学 2017-01-11 CN disclosed