SCHEMBL28119075

SCHEMBL28119075

Cc1ccc(-c2ccsc2C(C)C)cc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.44
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
HSD17B10 Q99714 1/20 0.35
PTGS1 P23219 4/20 0.34
LDHA P00338 1/20 0.34
LDHB P07195 1/20 0.34
EDNRB P24530 1/20 0.33
EDNRA P25101 1/20 0.33
MAPK14 Q16539 1/20 0.33
MEN1 O00255 2/20 0.32
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
KMT2A Q03164 2/20 0.32
ACHE P22303 1/20 0.32
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9910776 0.82 BCAT2 (0.43) PTGS2ALDH1A1HSD17B10MEN1KMT2A
SCHEMBL6918591 0.79 AKR1C3 (0.46) PTGS2ALDH1A1MAPTTSHRMAPK1
SCHEMBL28119077 0.78 ALDH1A1 (0.44) ALDH1A1MAPTHSD17B10LDHALDHB
SCHEMBL8089263 0.74 PTGS2 (0.49) PTGS2ALDH1A1MAPTTSHRMAPK1
SCHEMBL28228496 0.72 PTGS2 (0.71) PTGS2PTGS1MAPK14
Ammonia Solution, Strong SCHEMBL23908216 0.71 PTGS2 (0.69) PTGS2PTGS1MAPK14
SCHEMBL2231313 0.71 ALDH1A1 (0.47) PTGS2ALDH1A1MAPTTSHRMAPK1
SCHEMBL2781156 0.71 PTGS2 (0.46) PTGS2ALDH1A1MAPTTSHRMAPK1
SCHEMBL827163 0.69
SCHEMBL3988930 0.68 PTGS2 (0.44) PTGS2ALDH1A1MAPTTSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106414443-B Pyridopyrimidine dione derivative 诺华股份有限公司 2018-10-26 CN claimed
CN-106414443-A Pyridopyrimidinedione derivatives 诺华股份有限公司 2017-02-15 CN claimed
CN-106414443-B Pyridopyrimidine dione derivative 诺华股份有限公司 2018-10-26 CN disclosed
CN-106414443-A Pyridopyrimidinedione derivatives 诺华股份有限公司 2017-02-15 CN disclosed