SCHEMBL28124282

SCHEMBL28124282

C=C(C(=O)OC(=O)c1c(CBr)cccc1[N+](=O)[O-])C(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
HTT P42858 1/20 0.40
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
NPSR1 Q6W5P4 1/20 0.35
MAOB P27338 1/20 0.34
KMT2A Q03164 1/20 0.34
LMNA P02545 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
POLB P06746 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28124773 0.83 TDP1 (0.55) ALDH1A1HTTTDP1L3MBTL1NPSR1
SCHEMBL17335022 0.81 TDP1 (0.42) ALDH1A1HTTTDP1L3MBTL1NPSR1
SCHEMBL283180 0.79 SMN1; SMN2 (0.47) ALDH1A1HTTTDP1L3MBTL1NPSR1
SCHEMBL27415134 0.79 PDK1 (0.41) ALDH1A1NPSR1KMT2ALMNASMN1; SMN2
SCHEMBL28124769 0.79 ALDH1A1 (0.39) ALDH1A1HTTTDP1L3MBTL1NPSR1
SCHEMBL27448923 0.79 KMT2A (0.40) ALDH1A1HTTNPSR1KMT2ALMNA
SCHEMBL28124280 0.78 TDP1 (0.37) ALDH1A1HTTTDP1L3MBTL1NPSR1
SCHEMBL1143703 0.77 ALDH1A1 (0.48) ALDH1A1TDP1L3MBTL1KMT2ALMNA
SCHEMBL27570720 0.76 ALDH1A1 (0.46) ALDH1A1HTTNPSR1KMT2ASMN1; SMN2
SCHEMBL27720989 0.75 GPR35 (0.46) ALDH1A1HTTTDP1NPSR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106459012-A Quinazolinone derivatives as phosphatidylinositol 3-kinase inhibitors 吉利德科学公司 2017-02-22 CN disclosed