SCHEMBL27415134

SCHEMBL27415134

C=C(C(=O)OC(=O)c1ccc(CBr)c([N+](=O)[O-])c1)C(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.41
VCAM1 P19320 1/20 0.41
ALDH1A1 P00352 4/20 0.38
HPGD P15428 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
KMT2A Q03164 3/20 0.38
MAPT P10636 3/20 0.38
MEN1 O00255 1/20 0.38
RECQL P46063 1/20 0.38
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
PKM P14618 1/20 0.37
CRHBP P24387 1/20 0.37
CRHR2 Q13324 1/20 0.37
LMNA P02545 1/20 0.37
KDM4E B2RXH2 1/20 0.37
POLB P06746 1/20 0.37
CYP1A2 P05177 1/20 0.36
THRB P10828 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27448923 0.91 KMT2A (0.40) VCAM1ALDH1A1HPGDNPSR1KMT2A
SCHEMBL27337266 0.82 PDK1 (0.37) PDK1VCAM1ALDH1A1HPGDNPSR1
SCHEMBL27332233 0.82 VCAM1 (0.38) PDK1VCAM1ALDH1A1HPGDNPSR1
SCHEMBL27832784 0.81 VCAM1 (0.55) VCAM1ALDH1A1HPGDNPSR1KMT2A
SCHEMBL28791798 0.81 ITGB1 (0.51) VCAM1ALDH1A1HPGDNPSR1KMT2A
SCHEMBL6953347 0.81 PDK1 (0.46) PDK1VCAM1ALDH1A1HPGDNPSR1
SCHEMBL27416551 0.80 TSHR (0.55) VCAM1ALDH1A1KMT2AMAPTMEN1
SCHEMBL1018568 0.79 VCAM1 (0.58) PDK1VCAM1ALDH1A1HPGDNPSR1
SCHEMBL28824451 0.79 ATM (0.42) VCAM1ALDH1A1HPGDNPSR1KMT2A
SCHEMBL28124282 0.79 ALDH1A1 (0.40) ALDH1A1NPSR1KMT2ALMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1117569-C Bicyclic fibrinogen antagonists SMITHKLINE BEECHAM CORP (US) 2003-08-13 CN disclosed
CN-1143323-A Bicyclic fibrinogen antagonists SMITHKLINE BEECHAM CORP (US) 1997-02-19 CN disclosed