SCHEMBL2812660

SCHEMBL2812660

O=C1OC(=O)c2c(C#Cc3cccnc3)cccc21

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 4/20 0.41
CYP2A6 P11509 6/20 0.41
CYP2C9 P11712 3/20 0.40
CYP2B6 P20813 3/20 0.40
CYP2C19 P33261 3/20 0.40
CYP2D6 P10635 3/20 0.40
CYP2E1 P05181 2/20 0.40
CYP3A4 P08684 2/20 0.40
AAK1 Q2M2I8 1/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2C8 P10632 1/20 0.39
CHRNB2 P17787 2/20 0.38
CHRNA4 P43681 2/20 0.38
FFAR1 O14842 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL108548 0.82 ALOX15 (0.43) GRM5CYP2C9CYP2C19CYP2D6CYP3A4
SCHEMBL29546502 0.82 ALOX15 (0.43) GRM5CYP2C9CYP2C19CYP2D6CYP3A4
SCHEMBL12814518 0.81 TDP1 (0.48)
SCHEMBL28740199 0.75 CA12 (0.44) GRM5CYP2C9CYP2C19CYP3A4CYP1A2
SCHEMBL2812659 0.72 GRM5 (0.43) GRM5CYP1A2
SCHEMBL2810259 0.72 CREBBP (0.39) CYP2C9CYP2C19CYP2D6CYP3A4CYP1A2
SCHEMBL2815384 0.72 ALDH1A1 (0.46) GRM5CYP1A2
SCHEMBL3796332 0.72 CYP2A6 (0.67) GRM5CYP2A6CYP2C9CYP2B6CYP2C19
SCHEMBL2710468 0.72 ALOX15 (0.41)
SCHEMBL2810822 0.71 TYMS (0.39) GRM5CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100240908-A1 ACETYLENE COMPOUND FUJIFILM CORPORATION (JP) 2010-09-23 US disclosed
EP-2202221-A1 ACETYLENE COMPOUND Fujifilm Corporation (JP) 2010-06-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100240908-A1 ACETYLENE COMPOUND NAT1, KATNA1, KAT2B GRM5 2797/4885CYP2A6 2596/4885CYP2C9 1564/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.