SCHEMBL28130409

SCHEMBL28130409

Fc1cccc(-c2ccnc(-c3cccc(F)c3)c2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 2/20 0.55
KMO O15229 2/20 0.53
KDM4E B2RXH2 2/20 0.51
MEN1 O00255 1/20 0.51
MAPT P10636 1/20 0.51
KMT2A Q03164 1/20 0.51
GRM5 P41594 2/20 0.49
PIM1 P11309 2/20 0.49
BCHE P06276 1/20 0.49
ACHE P22303 1/20 0.49
IDO1 P14902 2/20 0.49
TAAR1 Q96RJ0 1/20 0.47
ESR2 Q92731 1/20 0.47
MAP4K4 O95819 2/20 0.46
CYP17A1 P05093 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP11B1 P15538 1/20 0.46
CYP11B2 P19099 1/20 0.46
FYN P06241 1/20 0.46
GABRG2 P18507 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27917353 0.93 CYP17A1 (0.57) MAPKAPK2KMOKDM4EMEN1MAPT
SCHEMBL25118560 0.90 IDO1 (0.55) MAPKAPK2KMOKDM4EMEN1MAPT
SCHEMBL4854402 0.83 GABRG2 (0.60) MAPKAPK2KMOPIM1GABRG2GABRB3
SCHEMBL842168 0.83 CYP2A6 (0.57) MAPKAPK2KMOKDM4EMEN1MAPT
SCHEMBL4227 0.83 KMO (0.49) MAPKAPK2KMOKDM4EMEN1MAPT
SCHEMBL25492416 0.83 KMO (0.49) MAPKAPK2KMOKDM4EMEN1MAPT
SCHEMBL27735978 0.82 MAP4K4 (0.53) MAPKAPK2KMOKDM4EMEN1MAPT
SCHEMBL14979564 0.81 ASIC3 (0.47) MAPKAPK2KMOGRM5IDO1TAAR1
SCHEMBL29398603 0.81 GRM5 (0.59) KMOKDM4EMEN1MAPTKMT2A
SCHEMBL2480128 0.81 GRM5 (0.59) KMOKDM4EMEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104822663-B Substituted N (3 (4 base of pyrimidine) phenyl) acrylamide as tyrosine receptor kinase BTK inhibitor is similar to thing 犹他大学研究基金会 2017-03-08 CN disclosed