SCHEMBL2814040

SCHEMBL2814040

COCCCn1c(C2CCCN(C(=O)C[C@@H](Cc3ccc(B4OC(C)(C)C(C)(C)O4)cc3)NC(=O)O)C2)cc2c(F)cccc21

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.34
REN P00797 7/20 0.32
ALDH1A1 P00352 1/20 0.32
TSHR P16473 1/20 0.32
KMT2A Q03164 1/20 0.32
CYP3A4 P08684 4/20 0.31
KCNH2 Q12809 1/20 0.31
HTR4 Q13639 1/20 0.31
ROCK1 Q13464 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2814043 1.00 CNR2 (0.34) CNR2RENALDH1A1TSHRKMT2A
SCHEMBL7898296 0.92 CNR2 (0.33) CNR2RENCYP3A4
SCHEMBL2790483 0.91 ALDH1A1 (0.31) RENALDH1A1TSHRKMT2A
SCHEMBL2790479 0.91 ALDH1A1 (0.31) RENALDH1A1TSHRKMT2A
SCHEMBL2790813 0.90 PROKR1 (0.36) CNR2ALDH1A1TSHRKMT2ACYP3A4
SCHEMBL2789237 0.89 CNR2 (0.37) CNR2RENALDH1A1TSHRKMT2A
SCHEMBL2789916 0.87 REN (0.32) RENALDH1A1TSHRKMT2ACYP3A4
SCHEMBL7902463 0.83 USP30 (0.33)
SCHEMBL7902090 0.83 USP30 (0.32) RENCYP3A4
SCHEMBL7897738 0.82 PADI4 (0.37) CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111634-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-30 WO disclosed