SCHEMBL28142804

SCHEMBL28142804

COC(=O)C[C@@]1(NC(=O)OC(C)(C)C)CCCC(F)(F)C1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.37
CA14 Q9ULX7 2/20 0.37
CA2 P00918 2/20 0.37
P2RX7 Q99572 1/20 0.34
CNR2 P34972 1/20 0.34
CTSL P07711 1/20 0.32
PPIA P62937 1/20 0.32
APLNR P35414 1/20 0.31
CTSK P43235 1/20 0.30
CYP2D6 P10635 1/20 0.30
CA1 P00915 1/20 0.30
CA7 P43166 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8282998 0.83 CA12 (0.42) CA12CA14CA2P2RX7CNR2
SCHEMBL13010604 0.81 CA2 (0.41) CA12CA14CA2P2RX7CNR2
SCHEMBL28142895 0.78 CA12 (0.36) CA12CA14CA2P2RX7CNR2
SCHEMBL22380429 0.76 CTSL (0.35) CA12CA14CA2P2RX7CTSL
SCHEMBL28143617 0.75 P2RX7 (0.35) CA12CA14CA2P2RX7CNR2
SCHEMBL3022379 0.75 CA12 (0.37) CA12CA14CA2P2RX7CNR2
SCHEMBL22633505 0.75 CA12 (0.36) CA12CA14CA2P2RX7CTSL
SCHEMBL6887591 0.74 APLNR (0.37) CA12CA14CA2P2RX7CTSL
SCHEMBL428722 0.74 P2RX7 (0.38) CA2P2RX7CTSLPPIAAPLNR
SCHEMBL25568153 0.74 CNR2 (0.37) CA12CA14CA2P2RX7CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104854087-B Indole carboxamide derivatives as P2X receptor antagonists 埃科特莱茵药品有限公司 2017-03-22 CN disclosed