SCHEMBL28145286

SCHEMBL28145286

NS(=O)(=O)c1cccc(-c2cncc(-c3ccsc3)c2)c1

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 7/20 0.58
CA2 P00918 7/20 0.58
CYP2A6 P11509 5/20 0.58
CA1 P00915 5/20 0.58
CA12 O43570 3/20 0.58
CHEK2 O96017 1/20 0.50
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2B6 P20813 1/20 0.46
CYP2C19 P33261 1/20 0.46
CDK8 P49336 1/20 0.46
LRRK2 Q5S007 2/20 0.45
KDR P35968 1/20 0.43
PTGES2 Q9H7Z7 1/20 0.43
CA13 Q8N1Q1 2/20 0.43
KAT6A Q92794 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31287798 0.90 CA2 (0.64) CA9CA2CYP2A6CA1CA12
SCHEMBL28145358 0.80 CYP2A6 (0.49) CA9CA2CYP2A6CA1CA12
SCHEMBL28844211 0.80 CDK8 (0.46) CA9CA2CA1CA12CDK8
SCHEMBL28844052 0.77 MAOA (0.60) CA9CA2CA1CA12CDK8
SCHEMBL11992658 0.77 MAOA (0.52) CA9CA2CA1CA12CDK8
SCHEMBL13035338 0.76 CYP2A6 (1.00) CYP2A6CHEK2CYP3A4CYP2C9CYP2B6
SCHEMBL2561753 0.74 CDK8 (0.48) CA9CA2CA1CA12CDK8
SCHEMBL14075569 0.74 CA9 (0.70) CA9CA2CYP2A6CA1CA12
SCHEMBL28145248 0.74 CA9 (0.64) CA9CA2CA1CA12CDK8
SCHEMBL28146304 0.74 CA9 (0.54) CA9CA2CA1CA12CDK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104334527-B Sulfonamide compounds and uses as tnap inhibitors 桑福德-伯纳姆医学研究院 2017-05-24 CN disclosed