SCHEMBL28148504

SCHEMBL28148504

CCC#Cc1cnccn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.47
HSP90AA1 P07900 1/20 0.33
CYP2C19 P33261 5/20 0.32
CYP2A6 P11509 5/20 0.32
CYP2D6 P10635 4/20 0.32
CYP2B6 P20813 4/20 0.32
CYP2C9 P11712 4/20 0.32
CYP2E1 P05181 3/20 0.32
CYP2C8 P10632 3/20 0.32
CYP19A1 P11511 1/20 0.32
POLB P06746 1/20 0.32
CHRNB2 P17787 2/20 0.31
CHRNA4 P43681 2/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
FGFR1 P11362 1/20 0.30
FGFR2 P21802 1/20 0.30
FGFR4 P22455 1/20 0.30
FGFR3 P22607 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17567286 0.84 GRM5 (0.45) GRM5HSP90AA1CYP2C19CYP2A6CYP2D6
SCHEMBL15870932 0.79 GRM5 (0.59) GRM5HSP90AA1POLBKDM4EHAO1
SCHEMBL31286309 0.79 GRM5 (0.59) GRM5HSP90AA1POLBKDM4EHAO1
SCHEMBL5240290 0.76 GRM5 (0.41) GRM5HSP90AA1POLBCHRNB2CHRNA4
SCHEMBL29994137 0.76
SCHEMBL15870983 0.76
SCHEMBL23583669 0.73 GRM5 (0.42) GRM5KDM4EALDH1A1SMN1; SMN2
SCHEMBL4637898 0.72 GRM5 (0.49) GRM5HSP90AA1KDM4EHAO1
SCHEMBL31036005 0.72 CHRNB2 (0.40) GRM5CYP2C19CYP2C9POLBCHRNB2
SCHEMBL29263693 0.72 CHRNB2 (0.40) GRM5CYP2C19CYP2C9POLBCHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106660994-A Phosphatidylinositol 3-kinase inhibitors 吉利德科学公司 2017-05-10 CN disclosed