SCHEMBL2814938

SCHEMBL2814938

CC1(C)OB(c2cnc(N)cc2F)OC1(C)C

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LPL P06858 1/20 0.34
LIPG Q9Y5X9 1/20 0.34
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
PDGFRB P09619 4/20 0.32
KDR P35968 4/20 0.32
EGFR P00533 2/20 0.32
CXCR2 P25025 1/20 0.31
AAK1 Q2M2I8 1/20 0.30
JAK2 O60674 1/20 0.30
BTK Q06187 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21828795 0.83 ABL1 (0.35) LPLLIPGPDGFRBKDR
SCHEMBL13016581 0.83 NOS3 (0.35) LPLLIPGNOS3NOS1NOS2
SCHEMBL13089602 0.81 NOS3 (0.47) NOS3NOS1NOS2PDGFRBKDR
SCHEMBL30736300 0.81 NOS3 (0.47) NOS3NOS1NOS2PDGFRBKDR
SCHEMBL2934443 0.80 PIK3R1 (0.38)
SCHEMBL5036984 0.80 LPL (0.34) LPLLIPGEGFRCXCR2JAK2
SCHEMBL29597659 0.80 EGFR (0.36) LPLLIPGEGFRCXCR2JAK2
SCHEMBL2818121 0.80 NOS3 (0.33) NOS3NOS1NOS2PDGFRBKDR
SCHEMBL16535156 0.80 EGFR (0.36) LPLLIPGEGFRCXCR2JAK2
Hydrochloric Acid SCHEMBL29960928 0.80 NOS3 (0.46) NOS3NOS1NOS2PDGFRBKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 36 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250340551-A1 SMALL MOLECULE MODULATORS OF STAT6 GILEAD SCIENCES INC (US) 2025-11-06 US disclosed
US-20240124467-A1 FUSED PYRIMIDINE COMPOUNDS AS INHIBITORS OF MENIN-MLL INTERACTION BIOMEA FUSION, INC. 2024-04-18 US disclosed
EP-4263542-A1 FUSED PYRIMIDINE COMPOUNDS AS INHIBITORS OF MENIN-MLL INTERACTION Biomea Fusion, Inc. (US) 2023-10-25 EP disclosed
WO-2022133064-A1 FUSED PYRIMIDINE COMPOUNDS AS INHIBITORS OF MENIN-MLL INTERACTION BIOMEA FUSION, INC. (US) 2022-06-23 WO disclosed
US-20140309221-A1 METHOD OF INHIBITING HAMARTOMA TUMOR CELLS DANA-FARBER CANCER INSTITUTE, INC. (US) 2014-10-16 US disclosed
US-20140309221-A1 METHOD OF INHIBITING HAMARTOMA TUMOR CELLS DANA-FARBER CANCER INSTITUTE, INC. (US) 2014-10-16 US disclosed
US-20140309221-A1 METHOD OF INHIBITING HAMARTOMA TUMOR CELLS DANA-FARBER CANCER INSTITUTE, INC. (US) 2014-10-16 US disclosed
EP-2673268-A1 METHOD OF INHIBITING HAMARTOMA TUMOR CELLS Dana-Farber Cancer Institute, Inc. (US) 2013-12-18 EP disclosed
US-8563549-B2 Pyrimidine derivatives used as PI-3 kinase inhibitors NOVARTIS AG (CH) 2013-10-22 US disclosed
US-8563549-B2 Pyrimidine derivatives used as PI-3 kinase inhibitors NOVARTIS AG (CH) 2013-10-22 US disclosed
EP-1984350-B1 PYRIMIDINE DERIVATIVES USED AS PI-3 KINASE INHIBITORS NOVARTIS AG (CH) 2010-08-18 EP disclosed
US-20100075965-A1 PI3 KINASE INHIBITORS AND METHODS OF THEIR USE NOVARTIS AG 2010-03-25 US disclosed
US-20100075965-A1 PI3 KINASE INHIBITORS AND METHODS OF THEIR USE NOVARTIS AG 2010-03-25 US disclosed
US-20100075965-A1 PI3 KINASE INHIBITORS AND METHODS OF THEIR USE NOVARTIS AG 2010-03-25 US disclosed
EP-1989201-A1 PI-3 KINASE INHIBITORS AND METHODS OF THEIR USE Novartis AG (CH) 2008-11-12 EP disclosed
EP-1984350-A1 PYRIMIDINE DERIVATIVES USED AS PI-3 KINASE INHIBITORS Novartis AG (CH) 2008-10-29 EP disclosed
WO-2007095588-A1 PI-3 KINASE INHIBITORS AND METHODS OF THEIR USE NOVARTIS AG (CH) 2007-08-23 WO disclosed
WO-2007095588-A1 PI-3 KINASE INHIBITORS AND METHODS OF THEIR USE NOVARTIS AG (CH) 2007-08-23 WO disclosed
WO-2007084786-A1 PYRIMIDINE DERIVATIVES USED AS PI-3 KINASE INHIBITORS NOVARTIS AG (CH) 2007-07-26 WO disclosed
WO-2007084786-A1 PYRIMIDINE DERIVATIVES USED AS PI-3 KINASE INHIBITORS NOVARTIS AG (CH) 2007-07-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250340551-A1 SMALL MOLECULE MODULATORS OF STAT6 STAT6, STAT1, STAT5B LPL 1257/4885LIPG 865/4885NOS3 884/4885
US-20240124467-A1 FUSED PYRIMIDINE COMPOUNDS AS INHIBITORS OF MENIN-MLL INTERACTION MLLT1, MEN1, MLLT3 LPL 4626/4885LIPG 4664/4885NOS3 4760/4885
US-20100075965-A1 PI3 KINASE INHIBITORS AND METHODS OF THEIR USE PIK3CA, PIK3CD, PIK3CB LPL 1484/4885LIPG 765/4885NOS3 3538/4885
US-20140309221-A1 METHOD OF INHIBITING HAMARTOMA TUMOR CELLS PHPT1, VHL, SDHA LPL 4236/4885LIPG 4749/4885NOS3 3328/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.