SCHEMBL28149706

SCHEMBL28149706

NC(=O)c1cnc(-c2cccnn2)s1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
GSK3B P49841 2/20 0.41
NPC1 O15118 5/20 0.41
RAB9A P51151 5/20 0.41
SMN1; SMN2 Q16637 4/20 0.41
MAPT P10636 2/20 0.41
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
LCK P06239 1/20 0.35
KCNH2 Q12809 1/20 0.35
ATM Q13315 1/20 0.35
P2RX7 Q99572 1/20 0.35
LIMK1 P53667 3/20 0.35
CHEK1 O14757 1/20 0.35
AURKA O14965 1/20 0.35
DAPK3 O43293 1/20 0.35
PRKD3 O94806 1/20 0.35
MAP4K4 O95819 1/20 0.35
PAK4 O96013 1/20 0.35
ABL1 P00519 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12571407 0.86 ALDH1A1 (0.50) ALDH1A1NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL12571410 0.82 ALDH1A1 (0.50) ALDH1A1GSK3BNPC1RAB9ASMN1; SMN2
SCHEMBL6609203 0.81 ALDH1A1 (0.72) ALDH1A1GSK3BNPC1RAB9ASMN1; SMN2
SCHEMBL30664409 0.81 ALDH1A1 (0.72) ALDH1A1GSK3BNPC1RAB9ASMN1; SMN2
SCHEMBL17065303 0.76 IKBKB (0.46) ALDH1A1NPC1RAB9AMAPTHDAC1
SCHEMBL15002894 0.76 ALDH1A1 (0.42) ALDH1A1GSK3BNPC1RAB9ASMN1; SMN2
SCHEMBL29548990 0.74 CYP3A4 (0.56) ALDH1A1GSK3BNPC1RAB9ASMN1; SMN2
SCHEMBL5392323 0.74 CYP3A4 (0.56) ALDH1A1GSK3BNPC1RAB9ASMN1; SMN2
SCHEMBL24176348 0.74 ALDH1A1 (0.45) ALDH1A1GSK3BNPC1RAB9ASMN1; SMN2
SCHEMBL29548925 0.73 ADORA3 (0.46) ALDH1A1GSK3BNPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107266419-A Specific amino pyridazine class, thing in combination, and its application method 赛特凯恩蒂克公司 2017-10-20 CN disclosed
CN-103002897-B Certain amino-pyridazines, compositions thereof, and methods of use thereof 赛特凯恩蒂克公司 2017-06-09 CN disclosed