SCHEMBL28154192

SCHEMBL28154192

O=C1C(=O)N(Cc2ccc(Cl)cc2)c2cccc(Br)c21

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 4/20 0.60
BCHE P06276 2/20 0.60
CES2 O00748 1/20 0.60
CHRM5 P08912 3/20 0.51
CHRM1 P11229 2/20 0.51
CHRM3 P20309 1/20 0.51
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA9 Q16790 1/20 0.48
ALDH1A1 P00352 4/20 0.47
ALDH2 P05091 3/20 0.47
ALDH3A1 P30838 3/20 0.47
ACHE P22303 4/20 0.47
APAF1 O14727 3/20 0.45
TP53 P04637 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
MAPT P10636 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15215035 0.88 ALDH1A1 (0.59) CES1BCHECES2CHRM5CHRM1
SCHEMBL961634 0.87 LMNA (0.53) CES1BCHECES2CHRM5CHRM1
SCHEMBL29460878 0.83 CASP3 (0.54) CHRM5CHRM1CHRM3CA12CA1
SCHEMBL4739205 0.83 CASP3 (0.54) CHRM5CHRM1CHRM3CA12CA1
SCHEMBL3860379 0.79 CA2 (0.56) CES1CHRM5CHRM1CHRM3CA12
SCHEMBL3027106 0.75 CES1 (1.00) CES1BCHECES2CHRM5CHRM1
SCHEMBL30967408 0.74 ALDH1A1 (0.61) CES1BCHECES2CHRM5CHRM1
SCHEMBL281789 0.73 CYP1B1 (0.55) CES1BCHECHRM5CHRM1CHRM3
SCHEMBL23145007 0.73 CES1 (0.38) CES1BCHECHRM5CHRM1CHRM3
SCHEMBL29811809 0.73 CES1 (0.38) CES1BCHECHRM5CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104829608-B A kind of cumarin thiazole indolone type compound and its preparation method and purposes 吉首大学 2017-06-30 CN disclosed