SCHEMBL28158482

SCHEMBL28158482

C(=NC1c2ccccc2-c2ccccc21)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
MAPT P10636 3/20 0.41
XBP1 P17861 1/20 0.41
G6PC1 P35575 1/20 0.37
ACHE P22303 2/20 0.37
BACE1 P56817 2/20 0.37
NOX1 Q9Y5S8 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
KDM4E B2RXH2 1/20 0.35
GRIN2D O15399 2/20 0.35
GRIN3B O60391 2/20 0.35
GRIN1 Q05586 2/20 0.35
GRIN2A Q12879 2/20 0.35
GRIN2B Q13224 2/20 0.35
GRIN2C Q14957 2/20 0.35
GRIN3A Q8TCU5 2/20 0.35
TAAR1 Q96RJ0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30389716 1.00 LMNA (0.44) LMNAL3MBTL1MAPTXBP1G6PC1
SCHEMBL29229485 0.81 CHRM5 (0.53) MAPTALDH1A1MAPK1KDM4EGRIN2D
SCHEMBL27991294 0.78 CHRM5 (0.38) LMNAL3MBTL1MAPTG6PC1ACHE
SCHEMBL28186169 0.77 MAOB (0.45) LMNAMAPTALDH1A1MAPK1KDM4E
SCHEMBL28186173 0.77 MAOB (0.45) LMNAMAPTALDH1A1MAPK1KDM4E
SCHEMBL27804939 0.74 GPR3 (0.37) ACHEALDH1A1BCHEGPR3HTR2A
SCHEMBL28355026 0.73 GPR3 (0.34) LMNAACHEALDH1A1TSHRMAPK1
SCHEMBL28355025 0.73 GPR3 (0.34) LMNAACHEALDH1A1TSHRMAPK1
Ammonia Solution, Strong SCHEMBL28186930 0.72 GPR3 (0.33) LMNAACHEALDH1A1TSHRMAPK1
SCHEMBL2042756 0.71 ALDH1A1 (0.46) LMNAL3MBTL1MAPTXBP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109136974-A One kind (sp containing C2)-N key compound preparation method 中国科学院上海有机化学研究所 2019-01-04 CN disclosed
CN-107531737-A Synthesis of desosamine 哈佛大学的校长及成员们 2018-01-02 CN disclosed
CN-106998685-A 14-membered ketolides and methods of making and using the same 哈佛大学的校长及成员们 2017-08-01 CN disclosed