SCHEMBL28159337

SCHEMBL28159337

FC(F)(F)COCc1ccncn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
GRM5 P41594 1/20 0.36
KCNH3 Q9ULD8 1/20 0.34
GRIN1 Q05586 3/20 0.33
GRIN2B Q13224 3/20 0.33
GABRA1 P14867 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33
GABRA5 P31644 1/20 0.33
GABRA3 P34903 1/20 0.33
GABRA2 P47869 1/20 0.33
HSP90AA1 P07900 1/20 0.32
SYK P43405 1/20 0.32
AURKB Q96GD4 1/20 0.32
INCENP Q9NQS7 1/20 0.32
LOXL2 Q9Y4K0 2/20 0.32
SCN9A Q15858 2/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.31
PDE5A O76074 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20233500 0.82 GRM5 (0.36) GRM5KCNH3GABRA1GABRG2GABRB3
SCHEMBL28267948 0.81 KCNH3 (0.36) GRM5KCNH3GRIN1GRIN2BGABRA1
SCHEMBL874832 0.76 SMN1; SMN2 (0.42) ALDH1A1SYKAURKBINCENPRAB9A
SCHEMBL28266378 0.76 NAMPT (0.39) GRM5KCNH3GABRA1GABRG2GABRB3
SCHEMBL18431119 0.76 GRM5 (0.43) GRM5KCNH3GRIN1GRIN2BGABRA1
SCHEMBL30960194 0.75 KCNH3 (0.38) KCNH3GRIN1GRIN2BHSP90AA1LOXL2
SCHEMBL28025302 0.75 KCNH3 (0.38) KCNH3GRIN1GRIN2BHSP90AA1LOXL2
Bromide SCHEMBL11114317 0.74 GRM5 (0.40) GRM5KCNH3GABRA1GABRG2GABRB3
SCHEMBL28159342 0.72 ALDH1A1 (0.35) ALDH1A1GABRA1GABRG2GABRB3GABRA3
SCHEMBL20002092 0.72 RORC (0.33) GRM5KCNH3GRIN1GRIN2BGABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105263923-B Pyrimidine compounds and their use as gamma secretase modulators 阿克图拉姆生命科学股份公司 2017-06-23 CN disclosed