SCHEMBL28267948

SCHEMBL28267948

FC(F)(F)OCc1ccncn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH3 Q9ULD8 1/20 0.36
GABRA1 P14867 2/20 0.35
GABRG2 P18507 2/20 0.35
GABRB3 P28472 2/20 0.35
GABRA5 P31644 2/20 0.35
GABRA3 P34903 2/20 0.35
GABRA2 P47869 2/20 0.35
HSP90AA1 P07900 1/20 0.34
SYK P43405 1/20 0.33
AURKB Q96GD4 1/20 0.33
INCENP Q9NQS7 1/20 0.33
PDE10A Q9Y233 1/20 0.33
GRIN1 Q05586 3/20 0.32
GRIN2B Q13224 3/20 0.32
GRM5 P41594 1/20 0.32
RORC P51449 1/20 0.32
P2RX7 Q99572 1/20 0.31
LOXL2 Q9Y4K0 2/20 0.30
CYP2D6 P10635 1/20 0.30
NAMPT P43490 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002092 0.82 RORC (0.33) KCNH3GABRA1GABRG2GABRB3GABRA5
SCHEMBL28159337 0.81 ALDH1A1 (0.37) KCNH3GABRA1GABRG2GABRB3GABRA5
SCHEMBL16886264 0.80 RORC (0.33) KCNH3GABRA1GABRG2GABRB3GABRA5
SCHEMBL18215020 0.79 CYP3A4 (0.32) KCNH3GABRA1GABRG2GABRB3GABRA5
SCHEMBL20233500 0.74 GRM5 (0.36) KCNH3GABRA1GABRG2GABRB3GABRA5
SCHEMBL30960194 0.74 KCNH3 (0.38) KCNH3HSP90AA1GRIN1GRIN2BP2RX7
SCHEMBL28025302 0.74 KCNH3 (0.38) KCNH3HSP90AA1GRIN1GRIN2BP2RX7
SCHEMBL1263106 0.74
SCHEMBL242763 0.74
SCHEMBL11003033 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109071488-B Substituted 1,2, 3-triazoles as NR 2B-selective NMDA modulators 詹森药业有限公司 2021-08-13 CN disclosed
CN-109071488-A Substituted 1,2,3- triazole is as NR2B- selective NMDA regulator 詹森药业有限公司 2018-12-21 CN disclosed