SCHEMBL28159341

SCHEMBL28159341

CC(C)c1nccc(COCC(F)(F)F)n1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 3/20 0.36
TRPV3 Q8NET8 5/20 0.33
ALDH1A1 P00352 2/20 0.33
CYP2C19 P33261 2/20 0.32
CYP17A1 P05093 1/20 0.32
CYP2C9 P11712 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
CNR2 P34972 1/20 0.32
PIK3CA P42336 1/20 0.31
MEN1 O00255 1/20 0.31
CYP1A2 P05177 1/20 0.31
KMT2A Q03164 1/20 0.31
HRH4 Q9H3N8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25588431 0.77 RXRA (0.39) AAK1MEN1KMT2AHRH4
SCHEMBL28159342 0.76 ALDH1A1 (0.35) ALDH1A1HDAC1HDAC6PIK3CA
SCHEMBL15999367 0.76 NUDT1 (0.42) AAK1CYP2C19CYP17A1CYP2C9CNR2
SCHEMBL16398534 0.76 NUDT1 (0.42) ALDH1A1PIK3CAMEN1KMT2AHRH4
SCHEMBL15274637 0.73 HRH4 (0.35) AAK1TRPV3HRH4
SCHEMBL28159759 0.72 RXRA (0.34) TRPV3ALDH1A1CYP2C19CYP2C9PIK3CA
SCHEMBL12190563 0.71 SORD (0.39) AAK1CYP1A2HRH4
SCHEMBL23542736 0.70 AAK1 (0.35) AAK1HRH4
SCHEMBL2632658 0.70 IDH1 (0.42) CYP2C19HRH4
SCHEMBL8819724 0.70 HRH4 (0.35) AAK1HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105263923-B Pyrimidine compounds and their use as gamma secretase modulators 阿克图拉姆生命科学股份公司 2017-06-23 CN disclosed