SCHEMBL28166349

SCHEMBL28166349

[CH2]c1cn(-c2nccs2)nn1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.34
LMNA P02545 2/20 0.33
GLA P06280 1/20 0.33
ALDH1A1 P00352 4/20 0.32
PPARG P37231 1/20 0.32
MAPK10 P53779 1/20 0.32
KMT2A Q03164 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
NCOR2 Q9Y618 1/20 0.32
POLB P06746 1/20 0.32
APEX1 P27695 1/20 0.32
RECQL P46063 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
HSD17B10 Q99714 2/20 0.31
TSHR P16473 1/20 0.31
NOS1 P29475 1/20 0.31
GAA P10253 2/20 0.31
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14692457 0.73 AKR1C3 (0.40) TDP1ALDH1A1PPARGMAPK10KMT2A
SCHEMBL15933318 0.71 ALDH1A1 (0.43) TDP1LMNAALDH1A1PPARGMAPK10
SCHEMBL15930178 0.68 ALDH1A1 (0.37) TDP1LMNAALDH1A1PPARGMAPK10
SCHEMBL3988944 0.67 LMNA (0.39) TDP1LMNAGLAALDH1A1POLB
SCHEMBL21379809 0.67 TDP1 (0.34) TDP1LMNAGLAALDH1A1POLB
SCHEMBL909646 0.65 KCNJ1 (0.46) TDP1LMNAGLAALDH1A1POLB
Bromide SCHEMBL18010906 0.64 KCNJ1 (0.45) TDP1LMNAGLAALDH1A1PPARG
SCHEMBL30061281 0.63 ALDH1A1 (0.40) TDP1LMNAGLAALDH1A1PPARG
SCHEMBL16547534 0.63 TDO2 (0.39) TDP1LMNAGLAALDH1A1PPARG
SCHEMBL1782525 0.63 ALDH1A1 (0.45) TDP1LMNAGLAALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103857681-B It is used as the new big ring of factor XI, plasma thromboplastin antecedent A inhibitor 百时美施贵宝公司 2017-07-14 CN disclosed