SCHEMBL28173190

SCHEMBL28173190

Cc1nc(-n2ccnn2)cnc1C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 1/20 0.37
NOTUM Q6P988 1/20 0.36
EGLN2 Q96KS0 3/20 0.33
HCRTR1 O43613 3/20 0.32
HCRTR2 O43614 3/20 0.32
KDM6B O15054 1/20 0.31
TET2 Q6N021 1/20 0.31
OGFOD1 Q8N543 1/20 0.31
TET1 Q8NFU7 1/20 0.31
EGLN1 Q9GZT9 1/20 0.31
HIF1AN Q9NWT6 1/20 0.31
MYC P01106 1/20 0.31
MAP3K5 Q99683 1/20 0.31
HCAR2 Q8TDS4 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16039381 0.75 HCRTR2 (0.43) NOTUMEGLN2HCRTR1HCRTR2MYC
SCHEMBL17768591 0.72 NOTUM (0.35) NOTUMHCRTR1HCRTR2MYCHCAR2
SCHEMBL29483818 0.71 ALDH1A1 (0.44) HCAR2ALDH1A1
SCHEMBL7940956 0.71 NOTUM (0.44) KCNJ1NOTUMEGLN2MAP3K5
SCHEMBL20774263 0.69 NOTUM (0.37) NOTUMHCRTR1HCRTR2HCAR2
SCHEMBL18588653 0.69 HCRTR1 (0.56) NOTUMEGLN2HCRTR1HCRTR2MYC
SCHEMBL30112052 0.68 HPGD (0.39) MYCHCAR2KDM4EALDH1A1MAPT
SCHEMBL7422568 0.68 HPGD (0.39) MYCHCAR2KDM4EALDH1A1MAPT
SCHEMBL18993134 0.68 LMNA (0.63) KCNJ1EGLN2TET2OGFOD1TET1
SCHEMBL19481007 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107106558-A Having a2AAminopyrazine compounds with antagonist properties 默沙东公司 2017-08-29 CN disclosed