SCHEMBL28411490

SCHEMBL28411490

Fc1ccc(Nc2ncnc3cc(N4CCNCC4)c(F)cc23)cc1Cl

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EGFR P00533 18/20 0.60
ERBB2 P04626 3/20 0.56
FBP1 P09467 2/20 0.56
AURKA O14965 1/20 0.56
INSR P06213 1/20 0.56
PDGFRB P09619 1/20 0.56
FLT4 P35916 1/20 0.56
KDR P35968 1/20 0.56
CLK1 P49759 1/20 0.56
EPHB4 P54760 1/20 0.56
TEK Q02763 1/20 0.56
AURKB Q96GD4 1/20 0.56
GRM1 Q13255 1/20 0.54
ERBB4 Q15303 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28407489 0.88 EGFR (0.76) EGFRERBB2FBP1AURKAINSR
SCHEMBL7475167 0.87 EGFR (0.51) EGFR
SCHEMBL7473037 0.83 SRC (0.49) EGFRERBB2PDGFRBKDR
SCHEMBL28397062 0.82 EGFR (0.68) EGFRERBB2ERBB4
SCHEMBL28182145 0.81 EGFR (0.51) EGFRERBB2FBP1AURKAINSR
SCHEMBL28403915 0.81 EGFR (0.74) EGFRERBB2FBP1AURKAINSR
SCHEMBL28181388 0.80 EGFR (0.56) EGFRERBB2FBP1AURKAPDGFRB
SCHEMBL7469491 0.77 HTT (0.56) AURKAAURKB
SCHEMBL4358041 0.77 EGFR (0.56) EGFRERBB2FBP1AURKAINSR
SCHEMBL29731422 0.76 EGFR (0.98) EGFRERBB2FLT4KDREPHB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107200715-B Quinazoline derivative and application thereof in preparation of antitumor drugs 陕西师范大学 2020-05-29 CN claimed
CN-107200715-B Quinazoline derivative and application thereof in preparation of antitumor drugs 陕西师范大学 2020-05-29 CN disclosed