SCHEMBL28185367

SCHEMBL28185367

CSc1c(-c2ccccc2)nc2c(Br)cccc2c1C(=O)O

nearest known ligand 0.67

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.67
CYP2C19 P33261 1/20 0.67
GAA P10253 2/20 0.57
CYP2C9 P11712 2/20 0.56
ALDH1A1 P00352 1/20 0.56
DHODH Q02127 9/20 0.54
TACR3 P29371 2/20 0.47
PDE10A Q9Y233 2/20 0.44
TSHR P16473 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C8 P10632 1/20 0.44
PTGFR P43088 1/20 0.42
LMNA P02545 1/20 0.42
SELPLG Q14242 1/20 0.37
PRNP P04156 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1581556 0.81 CYP2D6 (1.00) CYP2D6CYP2C19GAACYP2C9ALDH1A1
Hydrochloric Acid SCHEMBL3326324 0.80 CYP2D6 (0.97) CYP2D6CYP2C19GAACYP2C9ALDH1A1
SCHEMBL18075786 0.78 ALDH1A1 (0.75) CYP2D6CYP2C19GAACYP2C9ALDH1A1
SCHEMBL2372698 0.69 DHODH (0.56) CYP2D6CYP2C19CYP2C9ALDH1A1DHODH
SCHEMBL28170815 0.69 DHODH (0.73) GAADHODHPDE10ATSHR
SCHEMBL17594326 0.69 PTGFR (0.55) DHODHTACR3PTGFR
SCHEMBL22734576 0.67 P2RX3 (0.45) GAAALDH1A1DHODHPDE10APRNP
SCHEMBL4228780 0.67 DHODH (0.70) GAADHODHPDE10ATSHR
SCHEMBL1581075 0.67 CYP2D6 (0.72) CYP2D6CYP2C19GAACYP2C9ALDH1A1
SCHEMBL20138876 0.67 PDE10A (0.40) GAAALDH1A1DHODHPDE10ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107428691-A Bicyclic formamides of 2 aryl quinoline 4 of substituted N and application thereof 拜耳制药股份公司 2017-12-01 CN disclosed