Isoquinoline

Isoquinoline

SCHEMBL28191817

NN1CC=Cc2ccccc21.c1ccc2cnccc2c1

nearest known ligand 0.33

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.33
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA9 Q16790 2/20 0.33
P2RX4 Q99571 1/20 0.33
CA14 Q9ULX7 1/20 0.33
CYP1A2 P05177 2/20 0.32
CYP3A4 P08684 2/20 0.32
CYP2C19 P33261 2/20 0.32
LMNA P02545 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
MAPT P10636 1/20 0.31
KDM4E B2RXH2 1/20 0.31
PRKD3 O94806 1/20 0.31
PRKCG P05129 1/20 0.31
PRKCB P05771 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
PRKCA P17252 1/20 0.31
PRKACA P17612 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4838385 0.81 LMNA (0.39) CA1CA2P2RX4CYP3A4LMNA
Isoquinoline SCHEMBL28191779 0.80 LMNA (0.40) P2RX4LMNAKDM4EROCK2ROCK1
Isoquinoline SCHEMBL28183569 0.80 HTT (0.33) P2RX4
Hydrochloric Acid SCHEMBL28248510 0.79 MAPK1 (0.38) P2RX4CYP3A4LMNA
Hydrochloric Acid SCHEMBL7448875 0.79 MAPK1 (0.38) P2RX4CYP3A4LMNA
Isoquinoline SCHEMBL28075529 0.79 P2RX4 (0.38) P2RX4CYP3A4LMNAROCK2ROCK1
Indole SCHEMBL28196583 0.72 TRPA1 (0.50) CA1CA2
Isoquinoline SCHEMBL28392791 0.71 CA1 (0.39) CA1CA2CYP1A2CYP3A4CYP2C19
Isoquinoline SCHEMBL1310260 0.71 CA1 (0.39) CA1CA2CYP1A2CYP3A4CYP2C19
Isoquinoline SCHEMBL1308876 0.71 CA1 (0.39) CA1CA2CYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108516974-A Amide compounds for the treatment of HIV 吉利德科学公司 2018-09-11 CN disclosed
CN-105705500-B Amide compounds for the treatment of HIV 吉利德科学公司 2018-05-29 CN disclosed
CN-105636953-B 1,4 dibasic pyridyl derivatives and its purposes for treating the illness related to SMN shortages 诺华股份有限公司 2018-01-02 CN disclosed