SCHEMBL4838385

SCHEMBL4838385

NN1CC=Cc2ccccc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.39
MAPK1 P28482 2/20 0.39
TSHR P16473 1/20 0.39
SCN4A P35499 1/20 0.39
SCN5A Q14524 1/20 0.39
SCN9A Q15858 1/20 0.39
P2RX4 Q99571 11/20 0.34
P2RX1 P51575 5/20 0.34
P2RX3 P56373 5/20 0.34
TLR9 Q9NR96 1/20 0.33
P2RX7 Q99572 3/20 0.32
CHRM2 P08172 1/20 0.31
HTR1A P08908 1/20 0.31
ADRA2A P08913 1/20 0.31
CHRM1 P11229 1/20 0.31
DRD2 P14416 1/20 0.31
ADRA2B P18089 1/20 0.31
ADRA2C P18825 1/20 0.31
DRD1 P21728 1/20 0.31
PTGS1 P23219 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7448875 0.98 MAPK1 (0.38) LMNAMAPK1TSHRSCN4ASCN5A
SCHEMBL29434173 0.76 P2RX4 (0.37) LMNAMAPK1TSHRSCN4ASCN5A
SCHEMBL1198914 0.76 P2RX4 (0.37) LMNAMAPK1TSHRSCN4ASCN5A
SCHEMBL4540872 0.74 MAPK1 (0.35) LMNAMAPK1TSHRSCN4ASCN5A
SCHEMBL2073989 0.74 MAPK1 (0.35) LMNAMAPK1TSHRSCN4ASCN5A
Iodide SCHEMBL7101346 0.74 P2RX4 (0.36) LMNAMAPK1TSHRSCN4ASCN5A
SCHEMBL374978 0.74 MAPK1 (0.39) LMNAMAPK1TSHRSCN4ASCN5A
SCHEMBL5213962 0.74 MAPK1 (0.35) LMNAMAPK1TSHRSCN4ASCN5A
SCHEMBL8857358 0.74 MAPK1 (0.35) LMNAMAPK1TSHRSCN4ASCN5A
SCHEMBL29506717 0.74 MAPK1 (0.39) LMNAMAPK1TSHRSCN4ASCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 55 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2950649-A2 AMINE COMPOUNDS HAVING ANTI-INFLAMMATORY, ANTIFUNGAL, ANTIPARASITIC AND ANTICANCER ACTIVITY Wellstat Therapeutics Corporation (US) 2015-12-09 EP claimed
WO-2014120995-A2 AMINE COMPOUNDS HAVING ANTI-INFLAMMATORY, ANTIFUNGAL, ANTIPARASITIC AND ANTICANCER ACTIVITY WELLSTAT THERAPEUTICS CORPORATION (US) 2014-08-07 WO claimed
CN-102216298-B Imidazopyridines and imidazopyrimidines as HIV-1 reverse transcriptase inhibitors CSIR INC 2014-04-16 CN claimed
CN-101061118-A Substituted bicyclic imidazo-3-ylamine compounds GRUENENTHAL GMBH (DE) 2007-10-24 CN claimed
WO-1999067238-A2 TETRAHYDROQUINOLINE-INDOLE DERIVATIVES ANTIMICROBIAL AGENTS, THEIR USES AND COMPOSITIONS CONTAINING THEM SEPRACOR, INC. (US) 1999-12-29 WO claimed
US-20250223261-A1 PROCESS FOR MAKING A TASTE-MODIFYING COMPOUND FIRMENICH SA (CH) 2025-07-10 US disclosed
US-20240101531-A1 PYRIDINAMINE DERIVATIVES AND THEIR USE AS POTASSIUM CHANNEL MODULATORS XENON PHARMACEUTICALS INC. (CA) 2024-03-28 US disclosed
US-20230390259-A1 PHARMACEUTICAL COMPOSITION COMPRISING PYRIDONE DERIVATIVES SK BIOPHARMACEUTICALS CO., LTD. (KR) 2023-12-07 US disclosed
WO-2023209143-A1 PROCESS FOR MAKING A TASTE-MODIFYING COMPOUND FIRMENICH SA (CH) 2023-11-02 WO disclosed
CN-114751903-B Nitrogen-containing fused heterocycle SHP2 inhibitor compound, preparation method and application 上海凌达生物医药有限公司 2023-09-15 CN disclosed
US-20210085658-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING PYRIDONE DERIVATIVES SK BIOPHARMACEUTICALS CO., LTD. 2021-03-25 US disclosed
US-10456385-B2 Pharmaceutical composition comprising pyridone derivatives SK BIOPHARMACEUTICALS CO., LTD. (KR) 2019-10-29 US disclosed
CN-1784231-A 1-amino 1H-imidazoquinolines 3M INNOVATIVE PROPERTIES CO (US) 2006-06-07 CN disclosed
WO-2003013523-A1 SH3 PROTEIN DOMAINS AND THEIR LIGANDS ADELAIDE RESEARCH & INNOVATION PTY LTD (AU) 2003-02-20 WO disclosed
EP-0470578-B1 Novel tricyclic compound or salts thereof, method for producing the same and antimicrobial agent containing the same WAKUNAGA SEIYAKU KK (JP) 1996-11-06 EP disclosed
US-5399553-A Oral absorbability WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1995-03-21 US disclosed
US-5254685-A Tricyclic compound or salts thereof, method for producing the same and antimicrobial agent containing the same WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1993-10-19 US disclosed
CN-1059144-A New tricyclic compound or its salt, prepare their method and contain their antiseptic-germicide WAKUNAGA SEIYAKU KK (JP) 1992-03-04 CN disclosed
EP-0470578-A1 Novel tricyclic compound or salts thereof, method for producing the same and antimicrobial agent containing the same WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1992-02-12 EP disclosed
WO-1990005523-A2 PHENANTHROLINEDICARBOXYLATE ESTERS, 4-AMINOQUINOLINE AND ISOQUINOLINE DERIVATIVES AS INHIBITORS OF HIV REVERSE TRANSCRIPTASE THE UPJOHN COMPANY (US) 1990-05-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250223261-A1 PROCESS FOR MAKING A TASTE-MODIFYING COMPOUND TAS2R4, TAS2R50, TAS2R60 LMNA 4091/4885MAPK1 1603/4885TSHR 4372/4885
US-20240101531-A1 PYRIDINAMINE DERIVATIVES AND THEIR USE AS POTASSIUM CHANNEL MODULATORS KCNA1, KCNB1, KCNB2 LMNA 739/4885MAPK1 720/4885TSHR 1321/4885
US-20230390259-A1 PHARMACEUTICAL COMPOSITION COMPRISING PYRIDONE DERIVATIVES PLPBP, PDXK, PIR LMNA 2543/4885MAPK1 1773/4885TSHR 3361/4885
US-10456385-B2 Pharmaceutical composition comprising pyridone derivatives PLPBP, PDXK, PIR LMNA 2543/4885MAPK1 1773/4885TSHR 3361/4885
US-20210085658-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING PYRIDONE DERIVATIVES PLPBP, PDXK, PNPO LMNA 2494/4885MAPK1 1666/4885TSHR 3392/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.