SCHEMBL28192083

SCHEMBL28192083

COC(=O)c1ccc(=O)n(C)c1Br

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.42
GAA P10253 3/20 0.42
GLA P06280 2/20 0.42
BRD4 O60885 1/20 0.41
CA12 O43570 2/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
CA7 P43166 2/20 0.41
CA9 Q16790 2/20 0.41
CA14 Q9ULX7 2/20 0.41
PDK2 Q15119 1/20 0.41
PDK4 Q16654 1/20 0.41
GABRA1 P14867 1/20 0.40
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40
GABRA3 P34903 1/20 0.40
NR4A2 P43354 2/20 0.40
ALDH1A1 P00352 5/20 0.39
LMNA P02545 3/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4142698 0.80 KDM4E (0.47) KDM4EGAAGLABRD4CA12
SCHEMBL28132837 0.79 KDM4E (0.42) KDM4EGAAGLABRD4CA12
SCHEMBL391606 0.79 ABL1 (0.49) KDM4EGAAGLABRD4CA12
SCHEMBL25308830 0.77 CA1 (0.43) KDM4EGAAGLABRD4CA12
SCHEMBL28267154 0.75 CA12 (0.41) KDM4EGAAGLABRD4CA12
SCHEMBL8380028 0.72 CA1 (0.52) KDM4EGAAGLACA12CA1
SCHEMBL3095482 0.71 TSHR (0.42) KDM4EGAABRD4GABRA1GABRG2
SCHEMBL28192085 0.71 SLC6A3 (0.50) KDM4EGAAGLABRD4GABRA1
SCHEMBL5231392 0.69 MYC (0.49) KDM4EGAAGLABRD4CA12
SCHEMBL3048628 0.69 GABRG2 (0.44) KDM4EGAAGLABRD4CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105745193-B Antimycotic oxo-dihydro pyridine carbohydrazide derivative 株式会社大熊制药 2017-12-01 CN disclosed