SCHEMBL28192141

SCHEMBL28192141

c1ccc(N2Cc3ccccc3N=C2c2cccnc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.54
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
CYP11B2 P19099 4/20 0.45
ALDH1A1 P00352 4/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNA5 P30532 1/20 0.40
CHRNA4 P43681 1/20 0.40
CDK5 Q00535 1/20 0.40
CDK5R1 Q15078 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
GAA P10253 1/20 0.39
CYP11B1 P15538 3/20 0.38
CYP1A2 P05177 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6258947 0.87 SIGMAR1 (0.65) SIGMAR1NPC1RAB9AALDH1A1MEN1
SCHEMBL28192755 0.85 CYP2A6 (0.41) SIGMAR1NPC1RAB9ACYP11B2ALDH1A1
SCHEMBL28192152 0.84 SIGMAR1 (0.58) SIGMAR1NPC1RAB9ACYP11B2ALDH1A1
SCHEMBL28324685 0.77 SIGMAR1 (0.53) SIGMAR1NPC1RAB9AALDH1A1KMT2A
SCHEMBL28324632 0.77 SIGMAR1 (0.53) SIGMAR1NPC1RAB9AL3MBTL1MEN1
SCHEMBL28561721 0.77 SIGMAR1 (0.56) SIGMAR1NPC1RAB9AHPGDSMN1; SMN2
SCHEMBL28192155 0.77 SIGMAR1 (0.56) SIGMAR1NPC1RAB9AALDH1A1KMT2A
SCHEMBL28192173 0.77 SIGMAR1 (0.56) SIGMAR1NPC1RAB9AMEN1KMT2A
SCHEMBL28854194 0.77 SIGMAR1 (0.52) SIGMAR1NPC1RAB9AHPGDSMN1; SMN2
SCHEMBL6040419 0.72 SIGMAR1 (0.54) SIGMAR1NPC1RAB9AHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107417628-A Diaryl quianzolinones, its preparation method and its medical usage and the pharmaceutical composition comprising such compound 中国人民解放军军事医学科学院毒物药物研究所 2017-12-01 CN claimed
CN-107417628-A Diaryl quianzolinones, its preparation method and its medical usage and the pharmaceutical composition comprising such compound 中国人民解放军军事医学科学院毒物药物研究所 2017-12-01 CN disclosed