SCHEMBL28192152

SCHEMBL28192152

c1ccc(N2Cc3ccccc3N=C2c2ccncc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.58
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
HPGD P15428 1/20 0.46
HRH4 Q9H3N8 1/20 0.38
LMNA P02545 2/20 0.38
NOTUM Q6P988 1/20 0.37
CDK5 Q00535 2/20 0.37
CDK5R1 Q15078 2/20 0.37
CCR3 P51677 1/20 0.37
CTSD P07339 1/20 0.37
EED O75530 1/20 0.36
ACHE P22303 2/20 0.36
BCHE P06276 1/20 0.36
CYP11B2 P19099 1/20 0.35
EGFR P00533 1/20 0.35
MEN1 O00255 1/20 0.35
USP2 O75604 1/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6258947 0.91 SIGMAR1 (0.65) SIGMAR1NPC1RAB9ASMN1; SMN2HPGD
SCHEMBL28192141 0.84 SIGMAR1 (0.54) SIGMAR1NPC1RAB9ASMN1; SMN2HPGD
SCHEMBL28561721 0.84 SIGMAR1 (0.56) SIGMAR1NPC1RAB9ASMN1; SMN2HPGD
SCHEMBL28192155 0.84 SIGMAR1 (0.56) SIGMAR1NPC1RAB9ASMN1; SMN2HPGD
SCHEMBL28192173 0.84 SIGMAR1 (0.56) SIGMAR1NPC1RAB9ASMN1; SMN2HPGD
SCHEMBL28324685 0.81 SIGMAR1 (0.53) SIGMAR1NPC1RAB9ASMN1; SMN2HPGD
SCHEMBL28324632 0.81 SIGMAR1 (0.53) SIGMAR1NPC1RAB9ASMN1; SMN2HPGD
SCHEMBL28192123 0.79 SIGMAR1 (0.38) SIGMAR1NPC1RAB9ASMN1; SMN2HPGD
SCHEMBL6040419 0.78 SIGMAR1 (0.54) SIGMAR1NPC1RAB9ASMN1; SMN2HPGD
SCHEMBL28854194 0.77 SIGMAR1 (0.52) SIGMAR1NPC1RAB9ASMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107417628-A Diaryl quianzolinones, its preparation method and its medical usage and the pharmaceutical composition comprising such compound 中国人民解放军军事医学科学院毒物药物研究所 2017-12-01 CN claimed
CN-107417628-A Diaryl quianzolinones, its preparation method and its medical usage and the pharmaceutical composition comprising such compound 中国人民解放军军事医学科学院毒物药物研究所 2017-12-01 CN disclosed