SCHEMBL28198655

SCHEMBL28198655

OCc1cncc(-c2ccn(O)n2)c1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 4/20 0.41
CYP11B1 P15538 2/20 0.41
CYP2A6 P11509 1/20 0.41
FYN P06241 10/20 0.39
DYRK1A Q13627 1/20 0.38
MKNK1 Q9BUB5 2/20 0.37
MKNK2 Q9HBH9 2/20 0.37
PRMT5 O14744 1/20 0.35
WDR77 Q9BQA1 1/20 0.35
S1PR1 P21453 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17247603 0.84 MKNK1 (0.52) CYP11B2CYP11B1CYP2A6FYNDYRK1A
SCHEMBL21634194 0.69 CYP2A6 (0.50) CYP2A6FYNMKNK1MKNK2
SCHEMBL28197944 0.69 PIK3CA (0.38) FYNDYRK1AS1PR1
SCHEMBL5021553 0.68 FDPS (0.57) CYP11B2CYP11B1CYP2A6MKNK1MKNK2
SCHEMBL28855820 0.68 CSNK1D (0.42) FYNS1PR1
SCHEMBL2728918 0.67 CYP2A6 (0.47) CYP11B2CYP11B1CYP2A6DYRK1AMKNK1
SCHEMBL28197938 0.67 P2RX7 (0.36) S1PR1
SCHEMBL8336937 0.67 CYP2A6 (0.54) CYP11B2CYP11B1CYP2A6DYRK1A
SCHEMBL18851872 0.66 FYN (0.42) FYN
SCHEMBL844549 0.66 MKNK1 (0.68) CYP11B2CYP11B1CYP2A6FYNDYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107667106-A 2 (base of Pyrazolopyridine 3) pyrimidine derivatives as JAK inhibitor 阿尔米雷尔有限公司 2018-02-06 CN disclosed